TargetNF-kappa-B essential modulator(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataEC50: 5.00E+3nMAssay Description:Inhibition of GST-IkB phosphorylation by TNF-alpha stimulated HeLa cell lysate (IP-IKKgamma)More data for this Ligand-Target Pair
TargetNF-kappa-B essential modulator(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 80nMAssay Description:Binding affinity to full-length human NEMO (1 to 419 residues) assessed as dissociation constantMore data for this Ligand-Target Pair
TargetNF-kappa-B essential modulator(Homo sapiens (Human))
Millennium Pharmaceuticals
Curated by ChEMBL
Millennium Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 190nMAssay Description:Binding affinity to full-length human NEMO (1 to 419 residues) assessed as dissociation constantMore data for this Ligand-Target Pair