Found 5 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1A/1B/1D/1F/2A/2B/2C/3A/3B/4/5A/5B/6/7'
Target5-hydroxytryptamine receptor 1A/1B/1D/1F/2A/2B/2C/3A/3B/4/5A/5B/6/7(Rattus norvegicus)
Solvay Duphar
Curated by ChEMBL
Solvay Duphar
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:The binding affinity was measured on 5-hydroxytryptamine receptor uptake receptor using [3H]- paroxetine as radioligand.More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A/1B/1D/1F/2A/2B/2C/3A/3B/4/5A/5B/6/7(Rattus norvegicus)
Solvay Duphar
Curated by ChEMBL
Solvay Duphar
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]- GR-65,630 binding to 5-hydroxytryptamine 3 receptor in rat brain cortical membranesMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A/1B/1D/1F/2A/2B/2C/3A/3B/4/5A/5B/6/7(Rattus norvegicus)
Solvay Duphar
Curated by ChEMBL
Solvay Duphar
Curated by ChEMBL
Affinity DataIC50: 220nMAssay Description:In vitro inhibition of Angiotensin I converting enzymeMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A/1B/1D/1F/2A/2B/2C/3A/3B/4/5A/5B/6/7(Rattus norvegicus)
Solvay Duphar
Curated by ChEMBL
Solvay Duphar
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:In vitro inhibition of Angiotensin I converting enzymeMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A/1B/1D/1F/2A/2B/2C/3A/3B/4/5A/5B/6/7(Rattus norvegicus)
Solvay Duphar
Curated by ChEMBL
Solvay Duphar
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity at serotonin 5-HT1-type site receptor in rat cortex by displacing [3H]5-HTMore data for this Ligand-Target Pair