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Found 6 Enz. Inhib. hit(s) with Target = 'Apolipoprotein(a)'
TargetApolipoprotein(a)(Human)
Eli Lilly

US Patent
LigandPNGBDBM544449((2S)-3-[3-[[Bis[[3-[(2S)-2-carboxy-2-[(3R)-pyrroli...)
Affinity DataIC50: <0.314nMAssay Description:The in vitro binding affinity of compounds to the intended target human Apo(a) protein is tested in a competitive binding assay. Human Apo(a) protein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApolipoprotein(a)(Human)
Eli Lilly

US Patent
LigandPNGBDBM544455(3-[3-[[bis[[3-[2-carboxy-2-[(3R)-pyrrolidin-3-yl]p...)
Affinity DataIC50: <0.314nMAssay Description:The in vitro binding affinity of compounds to the intended target human Apo(a) protein is tested in a competitive binding assay. Human Apo(a) protein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApolipoprotein(a)(Human)
Eli Lilly

US Patent
LigandPNGBDBM544456((2S)-3-[3-[3-[(2S)-2-Carboxy-2-[(3R)-pyrrolidin-3-...)
Affinity DataIC50: <0.314nMAssay Description:The in vitro binding affinity of compounds to the intended target human Apo(a) protein is tested in a competitive binding assay. Human Apo(a) protein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApolipoprotein(a)(Human)
Eli Lilly

US Patent
LigandPNGBDBM544454((2S)-3-[3-[[[3-[(2S)-2-Carboxy-2-[(3R)-pyrrolidin-...)
Affinity DataIC50:  2.13nMAssay Description:The in vitro binding affinity of compounds to the intended target human Apo(a) protein is tested in a competitive binding assay. Human Apo(a) protein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApolipoprotein(a)(Human)
Eli Lilly

US Patent
LigandPNGBDBM544458((2R)-3-Phenyl-2-[(3S)-pyrrolidin-3-yl]propanoic ac...)
Affinity DataIC50:  126nMAssay Description:The in vitro binding affinity of compounds to the intended target human Apo(a) protein is tested in a competitive binding assay. Human Apo(a) protein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetApolipoprotein(a)(Human)
Eli Lilly

US Patent
LigandPNGBDBM544457((2S)-3-Phenyl-2-[(3R)-pyrrolidin-3-yl]propanoic ac...)
Affinity DataIC50:  152nMAssay Description:The in vitro binding affinity of compounds to the intended target human Apo(a) protein is tested in a competitive binding assay. Human Apo(a) protein...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent