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Found 262 Enz. Inhib. hit(s) with Target = 'Chymotrypsin-C'
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM87059(CHEMBL247767 | Chymostatin)
Affinity DataKi:  9.36nMAssay Description:inhibitory activity against alpha chymotrypsin from bovine pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM87059(CHEMBL247767 | Chymostatin)
Affinity DataKi:  9.36nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098882(4-[2-(5-Amino-6-oxo-2-m-tolyl-6H-pyrimidin-1-yl)-a...)
Affinity DataKi:  12.6nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50068918((S)-4-((2S,3S)-2-Benzyloxycarbonylamino-3-methyl-p...)
Affinity DataKi:  34nMAssay Description:Compound was evaluated for inhibitory activity against Bovine ChymotrypsinogenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50036127(CHEMBL11391 | {2-Oxo-6-phenyl-1-[(3,3,3-trifluoro-...)
Affinity DataKi:  55nMAssay Description:The compound was evaluated for the binding affinity against bovine pancreatic chymotrypsinogenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50036127(CHEMBL11391 | {2-Oxo-6-phenyl-1-[(3,3,3-trifluoro-...)
Affinity DataKi:  55nMAssay Description:Tested for inhibitory activity against bovine pancreatic chymotrypsinogenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM113119(US9695194, 6)
Affinity DataKi: <100nM ΔG°: <-41.6kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Chymotrypsin, bovine, 25 ug (Roche, sequence grade), Substrate S-2586 (Chromogenics, cat. no. 82 08 94). Chymotrypsin activity was determi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM113248(US9695194, 7)
Affinity DataKi: <100nM ΔG°: <-41.6kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Chymotrypsin, bovine, 25 ug (Roche, sequence grade), Substrate S-2586 (Chromogenics, cat. no. 82 08 94). Chymotrypsin activity was determi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM113283(US9695194, 8)
Affinity DataKi: <100nM ΔG°: <-41.6kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Chymotrypsin, bovine, 25 ug (Roche, sequence grade), Substrate S-2586 (Chromogenics, cat. no. 82 08 94). Chymotrypsin activity was determi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM113296(US9695194, 13)
Affinity DataKi: <100nM ΔG°: <-41.6kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Chymotrypsin, bovine, 25 ug (Roche, sequence grade), Substrate S-2586 (Chromogenics, cat. no. 82 08 94). Chymotrypsin activity was determi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM113300(US9695194, 16)
Affinity DataKi: <100nM ΔG°: <-41.6kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Chymotrypsin, bovine, 25 ug (Roche, sequence grade), Substrate S-2586 (Chromogenics, cat. no. 82 08 94). Chymotrypsin activity was determi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM113299(US9695194, 15)
Affinity DataKi: <100nM ΔG°: <-41.6kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Chymotrypsin, bovine, 25 ug (Roche, sequence grade), Substrate S-2586 (Chromogenics, cat. no. 82 08 94). Chymotrypsin activity was determi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM113297(US9695194, 14)
Affinity DataKi: <100nM ΔG°: <-41.6kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Chymotrypsin, bovine, 25 ug (Roche, sequence grade), Substrate S-2586 (Chromogenics, cat. no. 82 08 94). Chymotrypsin activity was determi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098877(4-{2-[5-Amino-2-(3-methoxy-phenyl)-6-oxo-6H-pyrimi...)
Affinity DataKi:  109nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098870(CHEMBL26182 | {4-[2-(5-Amino-6-oxo-2-m-tolyl-6H-py...)
Affinity DataKi:  147nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50061024((2-Methyl-1-{(S)-oxo-[(S)-2-((S)-3,3,3-trifluoro-1...)
Affinity DataKi:  149nMAssay Description:Binding affinity of the compound for human pancreatic ChymotrypsinogenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098884(4-[2-(5-Amino-6-oxo-2-pyridin-3-yl-6H-pyrimidin-1-...)
Affinity DataKi:  171nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098886(4-[2-(5-Amino-6-oxo-2-phenyl-6H-pyrimidin-1-yl)-ac...)
Affinity DataKi:  177nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM113293(US9695194, 10)
Affinity DataKi:  200nM ΔG°:  -39.8kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Chymotrypsin, bovine, 25 ug (Roche, sequence grade), Substrate S-2586 (Chromogenics, cat. no. 82 08 94). Chymotrypsin activity was determi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098885(4-[2-(5-Amino-6-oxo-2-pyridin-4-yl-6H-pyrimidin-1-...)
Affinity DataKi:  240nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50025549(6-Chloro-3-phenyl-pyran-2-one | CHEMBL274455)
Affinity DataKi:  270nMAssay Description:In vitro binding affinity towards alpha-chymotrypsin from bovine pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098866(4-({4-[2-(5-Amino-6-oxo-2-m-tolyl-6H-pyrimidin-1-y...)
Affinity DataKi:  282nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098883(4-[2-(5-Amino-6-oxo-2-m-tolyl-6H-pyrimidin-1-yl)-a...)
Affinity DataKi:  295nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098876(4-{2-[5-Amino-2-(3-fluoro-phenyl)-6-oxo-6H-pyrimid...)
Affinity DataKi:  306nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098871(4-[2-(5-Amino-6-oxo-2-m-tolyl-6H-pyrimidin-1-yl)-a...)
Affinity DataKi:  348nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50068894(3-(4-{[(S)-1-((S)-2-tert-Butoxycarbonylamino-3-met...)
Affinity DataKi:  364nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50068911(3-(4-{[(S)-1-(2-tert-Butoxycarbonylamino-3-methyl-...)
Affinity DataKi:  364nMAssay Description:Compound was evaluated for inhibitory activity against Bovine ChymotrypsinogenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM113292(US9695194, 9)
Affinity DataKi:  400nM ΔG°:  -38.0kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Chymotrypsin, bovine, 25 ug (Roche, sequence grade), Substrate S-2586 (Chromogenics, cat. no. 82 08 94). Chymotrypsin activity was determi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098889(4-[2-(5-Amino-6-oxo-2-m-tolyl-6H-pyrimidin-1-yl)-a...)
Affinity DataKi:  451nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098888(2-(5-Amino-6-oxo-2-m-tolyl-6H-pyrimidin-1-yl)-N-(1...)
Affinity DataKi:  455nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098874(4-{2-[5-Amino-2-(3-chloro-phenyl)-6-oxo-6H-pyrimid...)
Affinity DataKi:  458nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50068914(5-{(S)-2-[1-Benzyl-3-(3-butylsulfamoyl-phenylcarba...)
Affinity DataKi:  476nMAssay Description:Compound was evaluated for inhibitory activity against Bovine ChymotrypsinogenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50037325(CHEMBL113261 | {6-(4-Chloro-phenyl)-2-oxo-1-[(3,3,...)
Affinity DataKi:  500nMAssay Description:Tested for inhibitory activity against bovine pancreatic chymotrypsinogenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM113295(US9695194, 12)
Affinity DataKi:  600nM ΔG°:  -36.9kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Chymotrypsin, bovine, 25 ug (Roche, sequence grade), Substrate S-2586 (Chromogenics, cat. no. 82 08 94). Chymotrypsin activity was determi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50037329(CHEMBL432442 | {2-Oxo-6-p-tolyl-1-[(3,3,3-trifluor...)
Affinity DataKi:  720nMAssay Description:Tested for inhibitory activity against bovine pancreatic chymotrypsinogenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098880(3-{4-[2-(5-Amino-6-oxo-2-m-tolyl-6H-pyrimidin-1-yl...)
Affinity DataKi:  780nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM113294(US9695194, 11)
Affinity DataKi:  1.00E+3nM ΔG°:  -35.6kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Chymotrypsin, bovine, 25 ug (Roche, sequence grade), Substrate S-2586 (Chromogenics, cat. no. 82 08 94). Chymotrypsin activity was determi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50068920(5-{(S)-2-[1-Benzyl-3,3-difluoro-2-oxo-3-(3-sulfamo...)
Affinity DataKi:  1.03E+3nMAssay Description:Compound was evaluated for inhibitory activity against Bovine ChymotrypsinogenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098881(4-[2-(5-Amino-6-oxo-2-m-tolyl-6H-pyrimidin-1-yl)-a...)
Affinity DataKi:  1.09E+3nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM113301(US9695194, 17)
Affinity DataKi:  1.20E+3nM ΔG°:  -35.2kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Chymotrypsin, bovine, 25 ug (Roche, sequence grade), Substrate S-2586 (Chromogenics, cat. no. 82 08 94). Chymotrypsin activity was determi...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50068913(5-{(S)-2-[1-Benzyl-3-(3-carbamoyl-phenylcarbamoyl)...)
Affinity DataKi:  1.22E+3nMAssay Description:Compound was evaluated for inhibitory activity against Bovine ChymotrypsinogenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50025557(6-Chloro-5-phenyl-pyran-2-one | CHEMBL16220)
Affinity DataKi:  1.30E+3nMAssay Description:In vitro binding affinity towards alpha-chymotrypsin from bovine pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50068919(3-(4-{[(S)-1-(2-tert-Butoxycarbonylamino-4-carboxy...)
Affinity DataKi:  1.30E+3nMAssay Description:Compound was evaluated for inhibitory activity against Bovine ChymotrypsinogenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098892(4-[2-(5-Amino-6-oxo-2-m-tolyl-6H-pyrimidin-1-yl)-a...)
Affinity DataKi:  1.40E+3nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098867(3-{4-[2-(5-Amino-6-oxo-2-m-tolyl-6H-pyrimidin-1-yl...)
Affinity DataKi:  1.43E+3nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098875(4-[2-(5-Amino-6-oxo-2-m-tolyl-6H-pyrimidin-1-yl)-a...)
Affinity DataKi:  1.44E+3nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098846(2-[5-Amino-2-(4-fluoro-phenyl)-6-oxo-6H-pyrimidin-...)
Affinity DataKi:  1.63E+3nMAssay Description:Inhibitory activity against alpha chymotrypsin from bovine pancreas.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098872(CHEMBL442146 | {4-[2-(5-Amino-6-oxo-2-m-tolyl-6H-p...)
Affinity DataKi:  1.83E+3nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098891(4-[2-(5-Amino-6-oxo-2-m-tolyl-6H-pyrimidin-1-yl)-a...)
Affinity DataKi:  1.92E+3nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsin-C(Homo sapiens (Human))
Welfide

Curated by ChEMBL
LigandPNGBDBM50098879(4-[2-(5-Amino-6-oxo-2-m-tolyl-6H-pyrimidin-1-yl)-a...)
Affinity DataKi:  1.96E+3nMAssay Description:In vitro inhibitory activity was determined against bovine pancreas chymotrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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