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Found 234 Enz. Inhib. hit(s) with Target = 'Coagulation factor XIII A chain'
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM50083725(CHEMBL3423195)
Affinity DataIC50:  4nMAssay Description:Inhibition of thrombin-activated F13-A (unknown origin) in plasma assessed as inhibition of fibrin clot formation after 7 mins by biotin incorporatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM50083722(CHEMBL3423198)
Affinity DataIC50:  4nMAssay Description:Inhibition of thrombin-activated F13-A (unknown origin) in plasma assessed as inhibition of fibrin clot formation after 7 mins by biotin incorporatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Rat)
Zedira

US Patent
LigandPNGBDBM577483(US11472838, Compound 5)
Affinity DataIC50:  8nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM50245478(CHEMBL4081588 | US11472838, Compound Ref. 25)
Affinity DataIC50: >10nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577540(US11472838, Compound Ref. 16)
Affinity DataIC50: >10nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577546(US11472838, Compound Ref. 21)
Affinity DataIC50: >10nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577537(US11472838, Compound Ref. 14)
Affinity DataIC50: >10nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577509(US11472838, Compound 27 | US11472838, Compound 31a...)
Affinity DataIC50:  10nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577484(US11472838, Compound 1a/b)
Affinity DataIC50:  11nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577511(US11472838, Compound 29 | US11472838, Compound 32a...)
Affinity DataIC50:  12nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577487(US11472838, Compound 4)
Affinity DataIC50:  13nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Crab-eating macaque)
Zedira

US Patent
LigandPNGBDBM577483(US11472838, Compound 5)
Affinity DataIC50:  15nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577512(US11472838, Compound 30)
Affinity DataIC50:  15nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Mouse)
Zedira

US Patent
LigandPNGBDBM577483(US11472838, Compound 5)
Affinity DataIC50:  15nMAssay Description:The most relevant off-targets are the transglutaminase isoenzymes especially tissue transglutaminase (TG2) because the enzyme is ubiquitously express...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Pig)
Zedira

US Patent
LigandPNGBDBM577483(US11472838, Compound 5)
Affinity DataIC50:  16nMAssay Description:The most relevant off-targets are the transglutaminase isoenzymes especially tissue transglutaminase (TG2) because the enzyme is ubiquitously express...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577483(US11472838, Compound 5)
Affinity DataIC50:  16nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577485(US11472838, Compound 2a/b)
Affinity DataIC50:  16nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577483(US11472838, Compound 5)
Affinity DataIC50:  16nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577488(US11472838, Compound 6)
Affinity DataIC50:  17nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Rat)
Zedira

US Patent
LigandPNGBDBM577483(US11472838, Compound 5)
Affinity DataIC50:  17nMAssay Description:The most relevant off-targets are the transglutaminase isoenzymes especially tissue transglutaminase (TG2) because the enzyme is ubiquitously express...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577506(US11472838, Compound 24a/b)
Affinity DataIC50:  18nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Mouse)
Zedira

US Patent
LigandPNGBDBM577483(US11472838, Compound 5)
Affinity DataIC50:  19nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Crab-eating macaque)
Zedira

US Patent
LigandPNGBDBM577483(US11472838, Compound 5)
Affinity DataIC50:  19nMAssay Description:The most relevant off-targets are the transglutaminase isoenzymes especially tissue transglutaminase (TG2) because the enzyme is ubiquitously express...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577486(US11472838, Compound 3)
Affinity DataIC50:  20nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577507(US11472838, Compound 25a/b)
Affinity DataIC50:  20nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577489(US11472838, Compound 7a/b)
Affinity DataIC50:  21nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577490(US11472838, Compound 8a/b)
Affinity DataIC50:  21nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Dog)
Zedira

US Patent
LigandPNGBDBM577483(US11472838, Compound 5)
Affinity DataIC50:  24nMAssay Description:The most relevant off-targets are the transglutaminase isoenzymes especially tissue transglutaminase (TG2) because the enzyme is ubiquitously express...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577483(US11472838, Compound 5)
Affinity DataIC50:  24nMAssay Description:The most relevant off-targets are the transglutaminase isoenzymes especially tissue transglutaminase (TG2) because the enzyme is ubiquitously express...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577511(US11472838, Compound 29 | US11472838, Compound 32a...)
Affinity DataIC50:  24nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577483(US11472838, Compound 5)
Affinity DataIC50:  24nMAssay Description:The most relevant off-targets are the transglutaminase isoenzymes especially tissue transglutaminase (TG2) because the enzyme is ubiquitously express...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577496(US11472838, Compound 14a/b)
Affinity DataIC50:  26nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577509(US11472838, Compound 27 | US11472838, Compound 31a...)
Affinity DataIC50:  27nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Dog)
Zedira

US Patent
LigandPNGBDBM577483(US11472838, Compound 5)
Affinity DataIC50:  28nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577547(US11472838, Compound 45a/b)
Affinity DataIC50:  35nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577510(US11472838, Compound 28)
Affinity DataIC50:  36nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM50420503(CHEMBL2086505)
Affinity DataIC50:  39nMAssay Description:Inhibition of thrombin activated human F13a by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577530(US11472838, Compound 39a/b)
Affinity DataIC50:  39nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577499(US11472838, Compound 17a/b)
Affinity DataIC50:  41nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577518(US11472838, Compound 36a/b)
Affinity DataIC50:  41nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577504(US11472838, Compound 22a/b)
Affinity DataIC50:  42nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577492(US11472838, Compound 10a/b)
Affinity DataIC50:  42nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577508(US11472838, Compound 26a/b)
Affinity DataIC50:  43nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577528(US11472838, Compound 38)
Affinity DataIC50:  47nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM50083726(CHEMBL3423194)
Affinity DataIC50:  48nMAssay Description:Inhibition of thrombin-activated F13-A (unknown origin) in plasma assessed as inhibition of fibrin clot formation after 7 mins by biotin incorporatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577494(US11472838, Compound 12a/b)
Affinity DataIC50:  51nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM50420457(CHEMBL2086890)
Affinity DataIC50:  51nMAssay Description:Inhibition of thrombin activated human F13a by fluorescent transamidation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM50083728(CHEMBL3423193)
Affinity DataIC50:  55nMAssay Description:Inhibition of thrombin-activated F13-A (unknown origin) in plasma assessed as inhibition of fibrin clot formation after 7 mins by biotin incorporatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577534(US11472838, Compound 42a/b)
Affinity DataIC50:  56nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCoagulation factor XIII A chain(Homo sapiens (Human))
University Of Leeds

Curated by ChEMBL
LigandPNGBDBM577549(US11472838, Compound Ref. 23)
Affinity DataIC50:  56nMAssay Description:FXIIIa activity has been determined using substrate A101 (Zedira GmbH, Darmstadt, Germany), which is based on the N-terminal dodecapeptide of α2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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