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Found 137 Enz. Inhib. hit(s) with Target = 'Histamine receptor H3'
TargetHistamine receptor H3(Dog)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM22541(Clobenpropit | N''-[(4-chlorophenyl)methyl]{[3-(1H...)
Affinity DataKi:  0.0800nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50442630(CHEMBL2441638)
Affinity DataKi:  0.390nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50443217(CHEMBL3087669)
Affinity DataKi:  0.400nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50442628(CHEMBL2441640)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50442627(CHEMBL2441641)
Affinity DataKi:  0.550nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50442629(CHEMBL2441639)
Affinity DataKi:  0.550nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50442626(CHEMBL2441642)
Affinity DataKi:  0.850nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50442632(CHEMBL2441636)
Affinity DataKi:  0.970nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50443216(CHEMBL3087667)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Dog)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50158595((4'-(3-((2R,5R)-2,5-dimethylpyrrolidin-1-yl)propox...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Dog)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50074629(4-[(1R,2R)-2-(5,5-Dimethyl-hex-1-ynyl)-cyclopropyl...)
Affinity DataKi:  1.32nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50443227(CHEMBL3087356)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50443226(CHEMBL3087357)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50434389(CHEMBL2387288)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50437067(CHEMBL2403550)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cell membranes after 1 hr by scin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50437067(CHEMBL2403550)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50443225(CHEMBL3087671)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50443224(CHEMBL3087670)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50442640(CHEMBL2441653)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50434405(CHEMBL2387306)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50434382(CHEMBL2387309)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Dog)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50139391((R)-4-(2-(2-(2-methylpyrrolidin-1-yl)ethyl)benzofu...)
Affinity DataKi:  3.89nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50443223(CHEMBL3087358)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50442631(CHEMBL2441637)
Affinity DataKi:  3.90nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50434401(CHEMBL2387314)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50443222(CHEMBL3087673)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM200837(2-[2-((2s,3's)-2-methyl-[1,3']bipyrrolidin...)
Affinity DataKi:  4.21nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Dog)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50158601(A-317920 | CHEMBL361355 | Furan-2-carboxylic acid ...)
Affinity DataKi:  4.27nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50262939(2-Methyl-3-(4-{[3-(1-pyrrolidinyl)propyl]oxy}pheny...)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in HEK293T cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50443221(CHEMBL3087668)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50434400(CHEMBL2387315)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50443220(CHEMBL3087359)
Affinity DataKi:  4.70nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50443219(CHEMBL3087672)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Dog)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM27213(4-[3-(4-cyclopropanecarbonylphenoxy)propyl]-1H-imi...)
Affinity DataKi:  5.75nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Dog)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM27213(4-[3-(4-cyclopropanecarbonylphenoxy)propyl]-1H-imi...)
Affinity DataKi:  5.75nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50434392(CHEMBL2387285)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM247467(US9453023, 26)
Affinity DataKi:  6.01nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM247449(US9453023, 8)
Affinity DataKi:  6.07nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM247453(US9453023, 12)
Affinity DataKi:  6.10nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50193199((S)-1-(2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl)-3...)
Affinity DataKi:  6.30nMAssay Description:Binding affinity to rhesus monkey histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM247455(US9453023, 14)
Affinity DataKi:  6.61nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Dog)
Abbott Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi:  6.76nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50442631(CHEMBL2441637)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM247462(US9453023, 21)
Affinity DataKi:  6.88nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50434387(CHEMBL2387290)
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from cloned rhesus monkey histamine H3 receptor transfected in CHO cells after 1 hr by scintillation coun...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM200827(2-[2-methyl-6-((2s,3's)-2-methyl-[1,3']bip...)
Affinity DataKi:  7.10nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50437068(CHEMBL2403549)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from recombinant rhesus monkey histamine H3 receptor transfected in CHO cell membranes after 1 hr by scin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50442625(CHEMBL2441643)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM50442624(CHEMBL2441635)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rhesus monkey histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine receptor H3(Macaca mulatta (Rhesus macaque))
Sanofi Us

Curated by ChEMBL
LigandPNGBDBM200831(2-[2-methyl-6-((2s,3's)-2-methyl-[1,3']bip...)
Affinity DataKi:  7.57nMAssay Description:Rhesus H3 radioligand binding assay was performed using rhesus H3 receptor membranes (prepared as described above), [3H]-Methylhistamine (Perkin Elme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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