TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.890nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.900nMAssay Description:Thromboxane A2 synthase inhibitory activity was measured from inhibition of thromboxane B2 production in human platelet microsomesMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 0.900nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of thromboxane synthase (TXA2) in human platelet microsomes [reduced formation of TXB2 from prostaglandin H2(PGH2)]More data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1.20nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1.5nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 1.80nMAssay Description:In vitro inhibition of TXB2 production by incubating prostaglandin H2 with human platelet microsomes.More data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 2nMAssay Description:Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.More data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of thromboxane synthasase in microsomal platelet preparationMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of the compound against thromboxane synthaseMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of thromboxane synthaseMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Rattus norvegicus)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 2nMAssay Description:The compound was tested in vitro for its inhibitory activity against thromboxane synthase A2 (TXA2)More data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Rattus norvegicus)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Tested for inhibition of thromboxane synthetase from spontaneously hypertensive ratsMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 2nMAssay Description:Tested for 50% inhibition of thromboxane synthase (TxS) in human platelets (in vitro)More data for this Ligand-Target Pair
TargetThromboxane-A synthase(Rattus norvegicus)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against the production of thromboxane B2 (TXB2) in glycogen-induced peritoneal cells of ratMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 2.30nMAssay Description:Inhibition of thromboxane A2 synthetase from human platelets by 1 uM of the compoundMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 2.60nMAssay Description:In vitro for inhibitory activity against thromboxane synthaseMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 2.60nMAssay Description:In vitro inhibition of thromboxane synthasase in microsomal platelet preparationMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 2.70nMAssay Description:In vitro for inhibitory activity against thromboxane synthaseMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 2.90nMAssay Description:Activity against TXA2 synthase in bovine platelet microsomeMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 3nMAssay Description:Inhibition of thromboxane TXA2 synthetase from human plateletsMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against thromboxane A2 synthetaseMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 3nMAssay Description:In vitro activity on thromboxane A2 synthase inhibition in gel filtered human platelets.More data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 3nMAssay Description:In vitro activity on thromboxane A2 synthase inhibition in gel filtered human platelets.More data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of thromboxane synthase from human platelets.More data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 3nMAssay Description:Compound was evaluated in vitro for the inhibition of Thromboxane synthase using [14C]-arachidonic acid as radioligandMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair
TargetThromboxane-A synthase(Homo sapiens (Human))
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
University Of Li&Eagrove;Ge
Curated by PDSP Ki Database
Affinity DataIC50: 3nMAssay Description:In vitro inhibition of Thromboxane A2 synthaseMore data for this Ligand-Target Pair