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Found 524 Enz. Inhib. hit(s) with Target = 'Tubulin beta chain'
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485941(CHEMBL2181004)
Affinity DataKi:  0.0460nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485945(CHEMBL2181003)
Affinity DataKi:  0.0585nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485942(CHEMBL2181002)
Affinity DataKi:  0.0637nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485950(CHEMBL2181009)
Affinity DataKi:  0.122nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485944(CHEMBL2181006)
Affinity DataKi:  0.127nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485943(CHEMBL2181001)
Affinity DataKi:  0.131nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485946(CHEMBL2181000)
Affinity DataKi:  0.143nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485947(CHEMBL2181008)
Affinity DataKi:  0.183nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485949(CHEMBL2180999)
Affinity DataKi:  0.198nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485948(CHEMBL2181007)
Affinity DataKi:  0.280nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50485940(CHEMBL2181005)
Affinity DataKi:  0.367nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to pig brain tubulinMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataKi:  2.18E+3nMAssay Description:Binding affinity against tubulin using [3H]colchicine as radioligandMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataKi:  5.75E+3nMAssay Description:Binding affinity against tubulin usingf [3H]-colchicine as radioligandMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50146019(steganacin)
Affinity DataKi:  1.05E+4nMAssay Description:Binding affinity against tubulin using [3H]colchicine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50146021(CHEMBL152714)
Affinity DataKi:  3.20E+4nMAssay Description:Binding affinity against tubulin using [3H]colchicine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50146017(CHEMBL152476)
Affinity DataKi:  1.00E+5nMAssay Description:Binding affinity against tubulin using [3H]colchicine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50146018(CHEMBL3349041)
Affinity DataKi:  1.78E+5nMAssay Description:Binding affinity against tubulin using [3H]colchicine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50146022(CHEMBL346865)
Affinity DataKi:  1.85E+5nMAssay Description:Binding affinity against tubulin using [3H]colchicine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50146018(CHEMBL3349041)
Affinity DataKi:  1.85E+5nMAssay Description:Binding affinity against tubulin usingf [3H]-colchicine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50146016(CHEMBL149525)
Affinity DataKi:  2.01E+5nMAssay Description:Binding affinity against tubulin using [3H]colchicine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50500878(CHEMBL3799906)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of porcine brain tubulin polymerization measured every 1 min for 60 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50500880(CHEMBL3799435)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of porcine brain tubulin polymerization measured every 1 min for 60 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50500879(CHEMBL3800118)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of porcine brain tubulin polymerization measured every 1 min for 60 mins by microplate reader analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataIC50:  6.70nMAssay Description:Inhibition of porcine brain tubulin polymerization measured every 1 min for 60 mins by microplate reader analysisMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataIC50:  130nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetric assayMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataIC50:  130nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataIC50:  130nMAssay Description:Inhibition of tubulin polymerization in porcine brainMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataIC50:  130nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetryMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataIC50:  130nMAssay Description:Inhibition of pig tubulin polymerization determined after 45 mins at 37 degC by turbidimetric analysisMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataIC50:  130nMAssay Description:Inhibition of porcine brain tubulin polymerizationMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50012278((2ALPHA,2''BETA,3BETA,4ALPHA,5BETA)-VINCALEUKOBLAS...)
Affinity DataIC50:  130nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetry analysisMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50500399(CHEMBL3746906)
Affinity DataIC50:  160nMAssay Description:Displacement of [3H]-colchicine from biotinylated porcine tubulin after 2 hrs by competitive binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50474288(CHEMBL112192)
Affinity DataIC50:  220nMAssay Description:In vitro inhibitory concentration required to displace [3H]colchicine from its binding site on tubulinMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50477251(CHEMBL429265)
Affinity DataIC50:  290nMAssay Description:Inhibition of porcine brain tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50477242(CHEMBL240468)
Affinity DataIC50:  290nMAssay Description:Inhibition of porcine brain tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  350nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetric assayMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  350nMAssay Description:In vitro inhibition of maximum porcine tubulin assembly rate after 20 min at 37 degrees CMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  350nMAssay Description:Inhibition of porcine brain tubulin polymerizationMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  350nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetry analysisMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  350nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetryMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  350nMAssay Description:Inhibition of pig tubulin polymerization determined after 45 mins at 37 degC by turbidimetric analysisMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50035218(CHEMBL61 | PODOFILOX | Podophyllinic acid lactone ...)
Affinity DataIC50:  350nMAssay Description:Inhibition of tubulin polymerization in porcine brainMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50482385(CHEMBL1210322)
Affinity DataIC50:  360nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50469121(CHEMBL1210876)
Affinity DataIC50:  360nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50469125(CHEMBL1210959)
Affinity DataIC50:  360nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50474300(CHEMBL116173)
Affinity DataIC50:  370nMAssay Description:In vitro inhibitory concentration required to displace [3H]colchicine from its binding site on TubulinMore data for this Ligand-Target Pair
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50482387(CHEMBL1209944)
Affinity DataIC50:  380nMAssay Description:Inhibition of pig brain tubulin polymerization after 30 mins by turbidimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50476049(CHEMBL219102)
Affinity DataIC50:  380nMAssay Description:Inhibition of tubulin polymerization in porcine brainMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
University Of Bradford

Curated by ChEMBL
LigandPNGBDBM50477244(CHEMBL237880)
Affinity DataIC50:  390nMAssay Description:Inhibition of porcine brain tubulin polymerizationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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