Compile Data Set for Download or QSAR
maximum 50k data
Found 542 Enz. Inhib. hit(s) with Target = 'Type-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor'
LigandPNGBDBM50469937(CHEMBL104493)
Affinity DataKi:  0.126nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50469896(CHEMBL326910)
Affinity DataKi:  0.316nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50469890(CHEMBL63072)
Affinity DataKi:  0.398nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50469939(CHEMBL323125)
Affinity DataKi:  0.398nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50228201(CHEMBL265084)
Affinity DataKi:  0.460nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50469901(GR-138950 | SAPRISARTAN)
Affinity DataKi:  0.501nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50469888(CHEMBL104667)
Affinity DataKi:  0.631nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50228201(CHEMBL265084)
Affinity DataKi:  0.740nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat uterusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50469892(CHEMBL107081)
Affinity DataKi:  0.794nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50469886(CHEMBL107006)
Affinity DataKi:  0.794nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50228204(CHEMBL405389)
Affinity DataKi:  0.850nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50469893(CHEMBL104418)
Affinity DataKi:  1nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50228203(CHEMBL262025)
Affinity DataKi:  1nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50469940(CHEMBL105887)
Affinity DataKi:  1nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50469897(CHEMBL104281)
Affinity DataKi:  1nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50228204(CHEMBL405389)
Affinity DataKi:  1.20nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat uterusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50469934(CHEMBL324196)
Affinity DataKi:  1.30nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50469935(CHEMBL62909)
Affinity DataKi:  1.30nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50469889(CHEMBL62553)
Affinity DataKi:  1.30nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50469938(CHEMBL322989)
Affinity DataKi:  1.30nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50236697(5-L-isoleucineangiotensin II | 5-isoleucine-angiot...)
Affinity DataKi:  1.40nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228198(CHEMBL414796)
Affinity DataKi:  1.5nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat uterusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228199(ANGIOTENSIN AMIDE | Angiotensinamide)
Affinity DataKi:  1.60nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50469887(CHEMBL107043)
Affinity DataKi:  1.60nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50228200(CHEMBL217516)
Affinity DataKi:  1.60nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50469899(CHEMBL107967)
Affinity DataKi:  1.60nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50228203(CHEMBL262025)
Affinity DataKi:  1.70nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat uterusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228198(CHEMBL414796)
Affinity DataKi:  1.80nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50236697(5-L-isoleucineangiotensin II | 5-isoleucine-angiot...)
Affinity DataKi:  1.90nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat uterusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50469891(CHEMBL322516)
Affinity DataKi:  2nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50469900(CHEMBL104252)
Affinity DataKi:  2nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50212650(CHEMBL89917)
Affinity DataKi:  2.10nMAssay Description:Tested for binding affinity by measuring displacement of [125I]-Sar1 Ile8 angiotensin II from rat adrenal cortical membranesMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50469884(CHEMBL293447)
Affinity DataKi:  2.5nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50469894(CHEMBL323315)
Affinity DataKi:  2.5nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50469933(CHEMBL323378)
Affinity DataKi:  2.5nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50212651(CHEMBL422954)
Affinity DataKi:  2.60nMAssay Description:Tested for binding affinity by measuring displacement of [125I]-Sar1 Ile8 angiotensin II from rat adrenal cortical membranesMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50469895(CHEMBL104626)
Affinity DataKi:  3.20nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50469941(CHEMBL292040)
Affinity DataKi:  3.20nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50469936(CHEMBL108115)
Affinity DataKi:  4nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50228199(ANGIOTENSIN AMIDE | Angiotensinamide)
Affinity DataKi:  5.5nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat uterusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228200(CHEMBL217516)
Affinity DataKi:  6.10nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat uterusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50212649(CHEMBL91507)
Affinity DataKi:  6.90nMAssay Description:Tested for binding affinity by measuring displacement of [125I]-Sar1 Ile8 angiotensin II from rat adrenal cortical membranesMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50212692(CHEMBL88142)
Affinity DataKi:  7nMAssay Description:Tested for binding affinity by measuring displacement of [125I]-Sar1 Ile8 angiotensin II from rat adrenal cortical membranesMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50469902(CHEMBL320326)
Affinity DataKi:  20nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50212691(CHEMBL330062)
Affinity DataKi:  29nMAssay Description:Tested for binding affinity by measuring displacement of [125I]-Sar1 Ile8 angiotensin II from rat adrenal cortical membranesMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)
Affinity DataKi:  32nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50469885(CHEMBL418811)
Affinity DataKi:  32nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50228202(CHEMBL368638)
Affinity DataKi:  53nMAssay Description:Tested for inhibition of radioligand [Sar1,Ile5,8]AII binding to angiotensin II receptor in rat uterusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50469898(CHEMBL322828)
Affinity DataKi:  100nMAssay Description:Tested for in vitro binding affinity against angiotensin II receptor of rat liverMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50003399(4'-(2-Butyl-4-chloro-5-hydroxymethyl-imidazol-1-yl...)
Affinity DataKi:  350nMAssay Description:Tested for the binding affinity using radioligand [125I]-Sar1 Ile8-AII in the rat adrenal capsular membranes (adrenal cortex)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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