TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: 501nMAssay Description:Binding affinity to CK1a1 (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: 650nMAssay Description:Binding affinity to CK1a1 (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of CK1 (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of CK1 (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of CK1 (unknown origin)More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: >6.92E+3nMAssay Description:Inhibition of CK1alpha1More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: 3.83E+4nMAssay Description:Inhibition of casein kinase 1Checked by AuthorMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: 3.83E+4nM ΔG°: -25.6kJ/moleT: 2°CAssay Description:Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: 6.07E+4nM ΔG°: -24.5kJ/moleT: 2°CAssay Description:Protein kinase C, cAMP dependent protein kinase, cGMP dependent protein kinase and myosin light chain kinase activity were measure under conditions d...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: 8.00E+4nMAssay Description:Inhibition of casein kinase 1Checked by AuthorMore data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of human CK1-alpha1More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of Ck1alpha1More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 0.660nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 0.710nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 0.739nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 0.860nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 0.940nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 0.941nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 0.949nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 0.960nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.02nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.04nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.06nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.20nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.23nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.30nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.42nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:CSNK1A1-inhibitory activity of compounds of the present invention in presence of 1 μM adenosine-tri-phosphate (ATP) was quantified employing the...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.66nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.66nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.66nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.68nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.69nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.69nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.73nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair
TargetCasein kinase I isoform alpha(Homo sapiens (Human))
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Christian-Albrechts University Of Kiel
Curated by ChEMBL
Affinity DataIC50: 1.80nMAssay Description:Recombinant fusion protein of N-terminal Glutathion-S-Transferase (GST) and full-length human CSNK1A1, expressed by baculovirus infected insect cells...More data for this Ligand-Target Pair