TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataKi: >1.00E+3nM ΔG°: >-34.2kJ/molepH: 7.0 T: 2°CAssay Description:PTP activity was assayed using p-nitrophenyl phosphate (pNPP) as a substrate in DMG buffer (50 mM DMG, pH 7.0, 1 mM EDTA, 150 mM NaCl, 2 mM DTT, 0.1 ...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of VHX (unknown origin) expressed in Escherichia coli using pNPP substrate after 5 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of VHX (unknown origin) expressed in Escherichia coli using pNPP substrate after 5 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of DUSP22 (unknown origin) pre-incubated for 20 mins followed by fluorescence substrate addition and measured after 120 mins by DiFMUP ass...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 2.25E+3nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 23(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 2.30E+3nMAssay Description:For selectivity studies, the PTPs, including LYP, mPTPA, SHP1-D1C, PTP1B, LMPTP, VHR, Laforin and PTPα-D1D2 were expressed and purified from E. ...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 23(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of VHZ (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 2.35E+3nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 2.79E+3nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of VHX (unknown origin) expressed in Escherichia coli using pNPP substrate after 5 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 3.02E+3nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 23(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of recombinant VHZ (unknown origin) using pNPP as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 5.55E+3nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 23(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of recombinant VHZ (unknown origin) using pNPP as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 8.05E+3nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 8.36E+3nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 8.39E+3nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
Affinity DataIC50: 8.90E+3nMAssay Description:inhibition of Homo sapiens (human) recombinant DUSP26 catalytic domain (61 to 211 amino acid residues) overexpressed in Escherichia coli BL21 (DE3) a...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 2(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 9.20E+3nMAssay Description:Antagonist activity at human PAC1 expressed in mouse HIN 3T3 cells assessed as inhibition of glucagon-induced cAMP accumulation preincubated for 30 m...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 23(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of VHZ (unknown origin)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: >1.00E+4nMpH: 7.0Assay Description:PTP activity was assayed using p-nitrophenyl phosphate (pNPP) as a substrate in 3,3-dimethylglutarate buffer (50 mM 3,3-dimethylglutarate, pH 7.0, 1 ...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 23(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 1.14E+4nMpH: 7.0Assay Description:Inhibition of VHZ (unknown origin) using pNPP as substrate at pH 7 at 25 degC by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of GST-tagged human recombinant JSP1More data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+4nMAssay Description:inhibition of Homo sapiens (human) recombinant DUSP26 catalytic domain (61 to 211 amino acid residues) overexpressed in Escherichia coli BL21 (DE3) a...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
Affinity DataIC50: 1.67E+4nMAssay Description:Inhibition of DUSP26 (unknown origin)-mediated p38 dephosphorylationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+4nMAssay Description:inhibition of Homo sapiens (human) recombinant DUSP26 catalytic domain (61 to 211 amino acid residues) overexpressed in Escherichia coli BL21 (DE3) a...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
Affinity DataIC50: 1.98E+4nMAssay Description:inhibition of Homo sapiens (human) recombinant DUSP26 catalytic domain (61 to 211 amino acid residues) overexpressed in Escherichia coli BL21 (DE3) a...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
Affinity DataIC50: 2.23E+4nMAssay Description:inhibition of Homo sapiens (human) recombinant DUSP26 catalytic domain (61 to 211 amino acid residues) overexpressed in Escherichia coli BL21 (DE3) a...More data for this Ligand-Target Pair
Affinity DataIC50: 2.51E+4nMAssay Description:inhibition of Homo sapiens (human) recombinant DUSP26 catalytic domain (61 to 211 amino acid residues) overexpressed in Escherichia coli BL21 (DE3) a...More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of JNK-stimulating phosphatase-1 (JSP-1)More data for this Ligand-Target Pair
TargetDual specificity protein phosphatase 22(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of recombinant VHX (unknown origin) using OMFP as substrate after 1 hr by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.63E+4nMAssay Description:inhibition of Homo sapiens (human) recombinant DUSP26 catalytic domain (61 to 211 amino acid residues) overexpressed in Escherichia coli BL21 (DE3) a...More data for this Ligand-Target Pair
Affinity DataIC50: 2.69E+4nMAssay Description:inhibition of Homo sapiens (human) recombinant DUSP26 catalytic domain (61 to 211 amino acid residues) overexpressed in Escherichia coli BL21 (DE3) a...More data for this Ligand-Target Pair
Affinity DataIC50: 3.02E+4nMAssay Description:inhibition of Homo sapiens (human) recombinant DUSP26 catalytic domain (61 to 211 amino acid residues) overexpressed in Escherichia coli BL21 (DE3) a...More data for this Ligand-Target Pair
Affinity DataIC50: 3.66E+4nMAssay Description:inhibition of Homo sapiens (human) recombinant DUSP26 catalytic domain (61 to 211 amino acid residues) overexpressed in Escherichia coli BL21 (DE3) a...More data for this Ligand-Target Pair