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Found 3 Enz. Inhib. hit(s) with Target = 'Synapsin-1'
TargetSynapsin-1(Bos taurus)
Tu Dortmund University

Curated by ChEMBL
LigandPNGBDBM23408(2-(3,4-dihydroxyphenyl)-3,5,6,7-tetrahydroxy-4H-ch...)
Affinity DataIC50:  150nMAssay Description:Inhibition of bovine brain synapsin-1 incubated for 1 hr by ATP-[gamma35S] binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynapsin-1(Bos taurus)
Tu Dortmund University

Curated by ChEMBL
LigandPNGBDBM50180856(CHEMBL3818384)
Affinity DataIC50:  500nMAssay Description:Inhibition of bovine brain synapsin-1 incubated for 1 hr by ATP-[gamma35S] binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynapsin-1(Bos taurus)
Tu Dortmund University

Curated by ChEMBL
LigandPNGBDBM7533((2R)-2-[[6-(benzylamino)-9-isopropyl-purin-2-yl]am...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of bovine brain synapsin-1 incubated for 1 hr by ATP-[gamma35S] binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed