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Found 271 Enz. Inhib. hit(s) with Target = 'Thermolysin'
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50474105(CHEMBL43341)
Affinity DataKi:  0.0680nMAssay Description:pKi value expresses binding affinity against thermolysin pKi = -logKi (where Ki is in mol/L)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50006111((ZFPLA) 2-[2-(2-Benzyloxycarbonylamino-3-phenyl-pr...)
Affinity DataKi:  0.0680nMAssay Description:Inhibitory constant against thermolysin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50474138(CHEMBL38873)
Affinity DataKi:  1.51nMAssay Description:pKi value expresses binding affinity against thermolysin pKi = -logKi (where Ki is in mol/L)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070927(CHEMBL3409520)
Affinity DataKi:  4.90nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070925(CHEMBL3409522)
Affinity DataKi:  5.30nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070926(CHEMBL3409521)
Affinity DataKi:  5.5nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070924(CHEMBL3409523)
Affinity DataKi:  5.80nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50006110((ZGPLA) 2-[2-(2-Benzyloxycarbonylamino-acetylamino...)
Affinity DataKi:  9.10nMAssay Description:Inhibitory constant against thermolysin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50474141(CHEMBL43176)
Affinity DataKi:  9.12nMAssay Description:pKi value expresses binding affinity against thermolysin pKi = -logKi (where Ki is in mol/L)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070937(CHEMBL3409510)
Affinity DataKi:  10nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50121452((S)-2-{(S)-2-[(Benzyloxycarbonylamino-methyl)-hydr...)
Affinity DataKi:  11nMAssay Description:Competitive inhibition of thermolysin evaluated using the substrate FAGLA (Sigma); Competitive binding observedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50474083(CHEMBL41348)
Affinity DataKi:  11nMAssay Description:pKi value expresses binding affinity against thermolysin pKi = -logKi (where Ki is in mol/L)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50321113(3-Phenyl-2-(trifluoromethyl)quinazolin-4(3H)-one |...)
Affinity DataKi:  11.5nMAssay Description:Inhibition of Bacillus thermoproteolyticus thermolysin after 15 mins by microplate fluorescence analysis in presence of 0.5 to 2 mM substrate FaGLaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070922(CHEMBL3409525)
Affinity DataKi:  12nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50474089(CHEMBL43228)
Affinity DataKi:  16.6nMAssay Description:pKi value expresses binding affinity against thermolysin pKi = -logKi (where Ki is in mol/L)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50474119(CHEMBL40208)
Affinity DataKi:  18.6nMAssay Description:pKi value expresses binding affinity against thermolysin pKi = -logKi (where Ki is in mol/L)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50396788(CHEMBL2172738)
Affinity DataKi:  19nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50474137(CHEMBL41500)
Affinity DataKi:  19.1nMAssay Description:pKi value expresses binding affinity against thermolysin pKi = -logKi (where Ki is in mol/L)More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50396788(CHEMBL2172738)
Affinity DataKi:  19.1nMAssay Description:Binding affinity to Bacillus thermoproteolyticus thermolysin by UV-VIS spectrophotometric analysis in presence of 2-furanacryloyl-Gly-Leu-NH2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070917(CHEMBL3409528)
Affinity DataKi:  24nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070931(CHEMBL3409516)
Affinity DataKi:  26nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50251742((3R,4R,5R,6S)-3,4,5-trihydroxy-6-methyl-tetrahydro...)
Affinity DataKi:  28nMAssay Description:Inhibitory constant against thermolysin.More data for this Ligand-Target Pair
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50474108(CHEMBL41289)
Affinity DataKi:  28.2nMAssay Description:pKi value expresses binding affinity against thermolysin pKi = -logKi (where Ki is in mol/L)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070938(CHEMBL3409509)
Affinity DataKi:  29nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50442257(CHEMBL2028192)
Affinity DataKi:  30nMAssay Description:Inhibition of Bacillus thermoproteolyticus thermolysin using FA-Fly-Leu-NH2 as substrate at pH 7.5 after 15 mins by Henderson plot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070923(CHEMBL3409524)
Affinity DataKi:  31nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50442257(CHEMBL2028192)
Affinity DataKi:  32nMAssay Description:Inhibition of Bacillus thermoproteolyticus thermolysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50422014(CHEMBL319299)
Affinity DataKi:  33.9nMAssay Description:pKi value expresses binding affinity against thermolysin pKi = -logKi (where Ki is in mol/L)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070933(CHEMBL3409514)
Affinity DataKi:  37nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070920(CHEMBL3409526)
Affinity DataKi:  40nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50121454((S)-2-[(Aminomethyl-diphenyl-silanyl)-methyl]-4-me...)
Affinity DataKi:  41nMAssay Description:Competitive inhibition of thermolysin evaluated using the substrate FAGLA (Sigma); Competitive binding observedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50121453(CHEMBL334233 | Sodium; (S)-2-[(S)-2-({dihydroxy-[(...)
Affinity DataKi:  41nMAssay Description:Competitive inhibition of thermolysin evaluated using the substrate FAGLA (Sigma); Competitive binding observedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070930(CHEMBL3409517)
Affinity DataKi:  43nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50474144(CHEMBL287732)
Affinity DataKi:  44.7nMAssay Description:pKi value expresses binding affinity against thermolysin pKi = -logKi (where Ki is in mol/L)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50422014(CHEMBL319299)
Affinity DataKi:  50nMAssay Description:Tested for binding affinity against ThermolysinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50006117((CLT) 2-{1-[1-Carboxy-2-(1H-indol-3-yl)-ethylcarba...)
Affinity DataKi:  50nMAssay Description:Inhibitory constant against thermolysin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50474113(CHEMBL289703)
Affinity DataKi:  52.5nMAssay Description:pKi value expresses binding affinity against thermolysin pKi = -logKi (where Ki is in mol/L)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070918(CHEMBL3559407)
Affinity DataKi:  54nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070934(CHEMBL3409513)
Affinity DataKi:  59nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070936(CHEMBL3409511)
Affinity DataKi:  60nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50474121(CHEMBL436544)
Affinity DataKi:  66.1nMAssay Description:pKi value expresses binding affinity against thermolysin pKi = -logKi (where Ki is in mol/L)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070935(CHEMBL3409512)
Affinity DataKi:  67nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070941(CHEMBL3409506)
Affinity DataKi:  69nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50474120(CHEMBL290692)
Affinity DataKi:  75.9nMAssay Description:pKi value expresses binding affinity against thermolysin pKi = -logKi (where Ki is in mol/L)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070932(CHEMBL3409515)
Affinity DataKi:  100nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50474139(CHEMBL41376)
Affinity DataKi:  181nMAssay Description:pKi value expresses binding affinity against thermolysin pKi = -logKi (where Ki is in mol/L)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070928(CHEMBL3409519)
Affinity DataKi:  189nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50474086(CHEMBL288359)
Affinity DataKi:  218nMAssay Description:pKi value expresses binding affinity against thermolysin pKi = -logKi (where Ki is in mol/L)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50070943(CHEMBL3409505)
Affinity DataKi:  219nMAssay Description:Inhibition of Bacillus thermoproteolyticus TLN using 2-furanacryloyl-Gly-Leu-NH2 substrate by biochemical assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThermolysin(Bacillus thermoproteolyticus)
University Of Marburg

Curated by ChEMBL
LigandPNGBDBM50321123(3-(Isopropylideneamino)-2,2-dimethyl-2,3-dihydroqu...)
Affinity DataKi:  243nMAssay Description:Inhibition of Bacillus thermoproteolyticus thermolysin after 15 mins by microplate fluorescence analysis in presence of 0.5 to 2 mM substrate FaGLaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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