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Found 13 Enz. Inhib. hit(s) with Target = 'Vitamin D3 receptor A'
TargetVitamin D3 receptor A(Danio rerio)
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50241974(CHEMBL4099875)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at zebrafish VDR LBD (156 to 453 residues) expressed in HEK293 EBNA cells harboring human CYP24-Tk-Luc plasmid assessed as induction...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor A(Danio rerio)
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50241975(CHEMBL4060864)
Affinity DataEC50: >100nMAssay Description:Agonist activity at zebrafish VDR LBD (156 to 453 residues) expressed in HEK293 EBNA cells harboring human CYP24-Tk-Luc plasmid assessed as induction...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor A(Danio rerio)
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50241976(CHEMBL4088053)
Affinity DataEC50: >100nMAssay Description:Agonist activity at zebrafish VDR LBD (156 to 453 residues) expressed in HEK293 EBNA cells harboring human CYP24-Tk-Luc plasmid assessed as induction...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor A(Danio rerio)
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50241977(CHEMBL4066758)
Affinity DataEC50: >100nMAssay Description:Agonist activity at zebrafish VDR LBD (156 to 453 residues) expressed in HEK293 EBNA cells harboring human CYP24-Tk-Luc plasmid assessed as induction...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor A(Danio rerio)
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50496699(CHEMBL3220716)
Affinity DataEC50:  1.20nMAssay Description:Agonist activity at zebrafish gal4-VDR LBD expressed in human MCF7 cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor A(Danio rerio)
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataEC50:  5.5nMAssay Description:Agonist activity at zebrafish gal4-VDR LBD expressed in human MCF7 cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair
TargetVitamin D3 receptor A(Danio rerio)
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50409927(CHEMBL2112315)
Affinity DataKd: >3.00E+4nMAssay Description:Binding affinity to zebrafish VDR LBD assessed as Kd for fluorescein-labeled SRC1 NR2 peptide binding by micro-scale thermophoresis methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor A(Danio rerio)
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50496700(CHEMBL3220717)
Affinity DataKd:  1.80E+3nMAssay Description:Agonist activity at zebrafish VDR LBD assessed as binding affinity to TAMRA-labeled SRC-1 peptide by fluorescence anisotropy assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor A(Danio rerio)
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50496701(CHEMBL3220718)
Affinity DataKd:  1.80E+3nMAssay Description:Agonist activity at zebrafish VDR LBD assessed as binding affinity to TAMRA-labeled SRC-1 peptide by fluorescence anisotropy assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor A(Danio rerio)
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50496701(CHEMBL3220718)
Affinity DataEC50:  0.25nMAssay Description:Agonist activity at zebrafish gal4-VDR LBD expressed in human MCF7 cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor A(Danio rerio)
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50496699(CHEMBL3220716)
Affinity DataKd:  3.30E+3nMAssay Description:Agonist activity at zebrafish VDR LBD assessed as binding affinity to TAMRA-labeled SRC-1 peptide by fluorescence anisotropy assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor A(Danio rerio)
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50200182((1S,3R,5Z,7E)-9,10-secocholesta-5,7,10(19)-triene-...)
Affinity DataKd:  1.20E+3nMAssay Description:Binding affinity to zebrafish VDR LBD assessed as Kd for fluorescein-labeled SRC1 NR2 peptide binding by micro-scale thermophoresis methodMore data for this Ligand-Target Pair
TargetVitamin D3 receptor A(Danio rerio)
Institute Of Genetics And Molecular And Cellular Biology (Igbmc)

Curated by ChEMBL
LigandPNGBDBM50496700(CHEMBL3220717)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at zebrafish gal4-VDR LBD expressed in human MCF7 cells by luciferase reporter gene based transactivation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed