Compile Data Set for Download or QSAR

Found 10 hits with Target = 'Serine/threonine-protein kinase Aurora-A' for non-null ΔH°   

CellSerine/threonine-protein kinase Aurora-A(Human)
Moffitt Cancer Center

SyringePNGBDBM87047(Bisanilinopyrimidine, 3h | Bisanilinopyrimidine in...)
ITC Data−TΔS°: -16.1kJ/mole ΔH°: -59kJ/mole
pH: 7.4 T: 25.00°C 
CellSerine/threonine-protein kinase Aurora-A(Human)
Moffitt Cancer Center

SyringePNGBDBM87048(Bisanilinopyrimidine, 1 | Bisanilinopyrimidine inh...)
ITC Data−TΔS°: -14.0kJ/mole ΔH°: -59kJ/mole
pH: 7.4 T: 25.00°C 
In DepthDetails Article
PubMed
CellSerine/threonine-protein kinase Aurora-A(Human)
Moffitt Cancer Center

SyringePNGBDBM87049(Bisanilinopyrimidine inhibitor, 3)
ITC Data−TΔS°: 23.0kJ/mole ΔH°: -13kJ/mole
pH: 7.4 T: 25.00°C 
In DepthDetails Article
PubMed
CellSerine/threonine-protein kinase Aurora-A(Human)
Moffitt Cancer Center

SyringePNGBDBM87050(Bisanilinopyrimidine, 6h | Bisanilinopyrimidine in...)
ITC Data−TΔS°: -17.9kJ/mole ΔH°: -59kJ/mole
pH: 7.4 T: 25.00°C 
In DepthDetails Article
PubMed
CellSerine/threonine-protein kinase Aurora-A(Human)
Moffitt Cancer Center

SyringePNGBDBM87051(Bisanilinopyrimidine, 6d | Bisanilinopyrimidine in...)
ITC Data−TΔS°: -5.07kJ/mole ΔH°: -46kJ/mole
pH: 7.4 T: 25.00°C 
In DepthDetails Article
PubMed
CellSerine/threonine-protein kinase Aurora-A(Human)
Moffitt Cancer Center

SyringePNGBDBM87052(Bisanilinopyrimidine, 6a | Bisanilinopyrimidine in...)
ITC Data−TΔS°: -25.9kJ/mole ΔH°: -71kJ/mole
pH: 7.4 T: 25.00°C 
In DepthDetails Article
PubMed
CellSerine/threonine-protein kinase Aurora-A(Human)
Moffitt Cancer Center

SyringePNGBDBM87053(Bisanilinopyrimidine, 3l | Bisanilinopyrimidine in...)
ITC Data−TΔS°: -25.9kJ/mole ΔH°: -71kJ/mole
pH: 7.4 T: 25.00°C 
In DepthDetails Article
PubMed
CellSerine/threonine-protein kinase Aurora-A(Human)
Moffitt Cancer Center

SyringePNGBDBM87054(Bisanilinopyrimidine, 6i | Bisanilinopyrimidine in...)
ITC Data−TΔS°: -17.0kJ/mole ΔH°: -63kJ/mole
pH: 7.4 T: 25.00°C 
In DepthDetails Article
PubMed
CellSerine/threonine-protein kinase Aurora-A(Human)
Moffitt Cancer Center

SyringePNGBDBM87055(Bisanilinopyrimidine, 6n | Bisanilinopyrimidine in...)
ITC Data−TΔS°: -25.9kJ/mole ΔH°: -67kJ/mole
pH: 7.4 T: 25.00°C 
In DepthDetails Article
PubMed
CellSerine/threonine-protein kinase Aurora-A(Human)
Moffitt Cancer Center

SyringePNGBDBM87056(VX680)
ITC Data−TΔS°: -8.94kJ/mole ΔH°: -50kJ/mole
pH: 7.4 T: 25.00°C 
Syringe InfoPC cidPC sid
In DepthDetails Article
PubMed
  • Reorder this table by ΔH°
  • Reorder this table by ΔS°
  • Reorder this table by pH
  • Reorder this table by T
  • Change energy unit to:  kcal/mol