Compile Data Set for Download or QSAR

Found 9 hits with Target = 'hiv-1 protease mutant, mdr-qm'   

CellHIV-1 Protease Mutant, MDR-QM(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM580(AG1776 | (4R)-3-[(2S,3S)-2-hydroxy-3-[(3-hydroxy-2...)
ITC DataΔG°: -13.7kcal/mole −TΔS°: -9.79kcal/mole ΔH°: -3.89kcal/mole logk: 1.10E+10
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease Mutant, MDR-QM(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM578((2S)-N-[(2S,4S,5S)-5-[2-(2,6-dimethylphenoxy)aceta...)
ITC DataΔG°: -12.8kcal/mole −TΔS°: -15.6kcal/mole ΔH°: 2.80kcal/mole logk: 2.50E+9
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease Mutant, MDR-QM(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM577(VX-478 | 141W94 | APV | BDBM50215393 | CHEMBL116 |...)
ITC DataΔG°: -11.6kcal/mole −TΔS°: -11.1kcal/mole ΔH°: -0.499kcal/mole logk: 3.20E+8
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease Mutant, MDR-QM(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM518(Viracept | CHEMBL584 | (3S,4aS,8aS)-N-tert-butyl-2...)
ITC DataΔG°: -11.0kcal/mole −TΔS°: -18.3kcal/mole ΔH°: 7.29kcal/mole logk: 1.20E+8
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease Mutant, MDR-QM(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM579(Kynostatin 272 | CHEMBL414640 | (4R)-N-tert-butyl-...)
ITC DataΔG°: -10.9kcal/mole −TΔS°: -10.9kcal/mole ΔH°: 0kcal/mole logk: 9.00E+7
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease Mutant, MDR-QM(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM520(ABT-538 | Norvir | CHEMBL163 | 1,3-thiazol-5-ylmet...)
ITC DataΔG°: -10.7kcal/mole −TΔS°: -14.0kcal/mole ΔH°: 3.29kcal/mole logk: 7.40E+7
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease Mutant, MDR-QM(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM517(Crixivan | CHEMBL115 | L-735, 524 | MK639 | Indina...)
ITC DataΔG°: -10.4kcal/mole −TΔS°: -16.8kcal/mole ΔH°: 6.39kcal/mole logk: 4.50E+7
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease Mutant, MDR-QM(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM519(SQV | Invirase | CHEMBL114 | Ro 31-8959 | Fortovas...)
ITC DataΔG°: -9.98kcal/mole −TΔS°: -18.5kcal/mole ΔH°: 8.49kcal/mole logk: 2.30E+7
pH: 5.0 T: 25.00°C 
CellHIV-1 Protease Mutant, MDR-QM(Human immunodeficiency virus type 1)
The Johns Hopkins University

SyringePNGBDBM581(4-{2-[(3R)-4-[2-(2-acetamido-3-methylbutanamido)-3...)
ITC DataΔG°: -7.59kcal/mole −TΔS°: -19.8kcal/mole ΔH°: 12.2kcal/mole logk: 4.10E+5
pH: 5.0 T: 25.00°C 
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