Affinity DataEC50: 10nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:In vitro agonistic activity against cAMP accumulation level in CHO cells expressing human beta-AR receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 30nMAssay Description:Inhibition of Rap1A-mediated geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 31nMAssay Description:Compound was tested for its intrinsic activity against beta adrenergic receptor of isolated guinea pig atrial pairsMore data for this Ligand-Target Pair
Affinity DataEC50: 77nMAssay Description:In vitro agonistic activity against cAMP accumulation level in CHO cells expressing human beta-AR receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 2.60E+3nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 6.00E+3nMAssay Description:Inhibition of H-Ras-mediated farnesylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+4nMAssay Description:Beta-adrenergic agonistic activity in guinea-pig atrium preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+4nMAssay Description:Beta-adrenergic agonistic activity in guinea-pig atrium preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+4nMAssay Description:Beta-adrenergic agonistic activity in guinea-pig atrium preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+4nMAssay Description:Beta-adrenergic agonistic activity in guinea-pig atrium preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+4nMAssay Description:Beta-adrenergic agonistic activity in guinea-pig atrium preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+4nMAssay Description:Inhibition of Rap1A-mediated geranylgeranylation expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+4nMAssay Description:Beta-adrenergic agonistic activity in guinea-pig atrium preincubated with phenoxybenzamine (12 uM) for 30 minMore data for this Ligand-Target Pair