Compile Data Set for Download or QSAR
maximum 50k data
Found 57 of ec50 for UniProtKB: P11229
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475448(CHEMBL195011)
Affinity DataEC50:  1.74nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475454(CHEMBL196218)
Affinity DataEC50:  4.79nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50064609(6-acetoxy-8-azonia-bicyclo[3.2.1]octane | Acetic a...)
Affinity DataEC50:  6.17nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475459(CHEMBL194008)
Affinity DataEC50:  6.46nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475443(CHEMBL364454)
Affinity DataEC50:  26.9nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50046728(1-Methyl-5-(3-methyl-[1,2,4]oxadiazol-5-yl)-1,2,3,...)
Affinity DataEC50:  32nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475458(CHEMBL194793)
Affinity DataEC50:  44.7nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475453(CHEMBL372536)
Affinity DataEC50:  50.1nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM46858(1-methyl-3,6-dihydro-2H-pyridine-5-carboxylic acid...)
Affinity DataEC50:  73nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475449(CHEMBL197092)
Affinity DataEC50:  79.4nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475450(CHEMBL194196)
Affinity DataEC50:  89.1nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475446(CHEMBL196151)
Affinity DataEC50:  93.3nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50228570(CHEMBL1788202)
Affinity DataEC50:  94nMAssay Description:Compound was tested for its potency against Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229049(CHEMBL351934)
Affinity DataEC50:  100nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Affinity DataEC50:  100nMAssay Description:Compound was tested for its potency against Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475457(CHEMBL373341)
Affinity DataEC50:  104nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Affinity DataEC50:  110nMAssay Description:In vitro muscarinic activity was measured on isolated guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229060(CHEMBL161007)
Affinity DataEC50:  130nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229056(CHEMBL349025)
Affinity DataEC50:  150nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229046(CHEMBL159273)
Affinity DataEC50:  200nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475442(CHEMBL194847)
Affinity DataEC50:  263nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229067(CHEMBL355824)
Affinity DataEC50:  320nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229062(CHEMBL422538)
Affinity DataEC50:  420nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229044(CHEMBL349066)
Affinity DataEC50:  620nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Affinity DataEC50:  620nMAssay Description:In vitro muscarinic activity was measured on isolated guinea pig urinary bladderMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229061(CHEMBL162134)
Affinity DataEC50:  720nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229066(CHEMBL350949)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229054(CHEMBL161748)
Affinity DataEC50:  1.28E+3nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229055(CHEMBL161670)
Affinity DataEC50:  1.46E+3nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475444(CHEMBL196219)
Affinity DataEC50:  1.99E+3nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50228575(CHEMBL108140)
Affinity DataEC50:  2.80E+3nMAssay Description:Compound was tested for its potency against Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475440(CHEMBL193698)
Affinity DataEC50:  4.36E+3nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475447(CHEMBL193642)
Affinity DataEC50:  4.46E+3nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475452(CHEMBL425911)
Affinity DataEC50:  5.01E+3nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50228578(CHEMBL111327)
Affinity DataEC50:  7.50E+3nMAssay Description:Compound was tested for its potency against Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475461(CHEMBL194144)
Affinity DataEC50:  1.14E+4nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50475441(CHEMBL62560)
Affinity DataEC50:  1.47E+4nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50064612(6-acetoxy-8-methyl-8-azonia-bicyclo[3.2.1]octane |...)
Affinity DataEC50:  2.45E+4nMAssay Description:Agonistic activity against Muscarinic acetylcholine receptor of guinea pig ileal longitudinal muscleMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229068(CHEMBL159311)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229045(CHEMBL159841)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229047(CHEMBL159628)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229065(CHEMBL262517)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229058(CHEMBL161088)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229064(CHEMBL159839)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229051(CHEMBL159935)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229052(CHEMBL159651)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229053(CHEMBL161364)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229059(CHEMBL159708)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229057(CHEMBL161419)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1/M2/M3/M4/M5(Homo sapiens (Human))
Shanghai Second Medical University

Curated by ChEMBL
LigandPNGBDBM50229050(CHEMBL422710)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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