Affinity DataEC50: 0.191nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 0.257nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 0.324nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 0.389nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 0.468nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 0.501nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 0.692nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 0.871nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 1.40nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 1.90nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 1.90nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 2.20nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 2.60nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.60nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.80nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 3.40nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 3.5nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 3.70nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 3.80nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 4.90nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 5.5nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 5.80nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 6.30nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 7.40nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 7.40nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 9.5nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 9.80nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 32nMAssay Description:Concentration required for coronary arteries vasodilation at the Adenosine A2 receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 35nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 51nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 62nMAssay Description:Concentration required for coronary arteries vasodilation at the A2 adenosine receptor in langendorff guinea pig heart preparationMore data for this Ligand-Target Pair
Affinity DataEC50: 62nMAssay Description:Binding affinity against Adenosine A2 receptor from rat striatal membranes with 50 nM CPA using [3H]-NECAMore data for this Ligand-Target Pair
Affinity DataEC50: 76nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 79nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 105nMAssay Description:Inhibition of adenylate cyclase via Adenosine A1 receptor in rat fat cell membranesMore data for this Ligand-Target Pair
Affinity DataEC50: 127nMAssay Description:Maximal NECA stimulation of adenylate cyclase via adenosine A2 receptor in human platelet membranesMore data for this Ligand-Target Pair
Affinity DataEC50: 128nMAssay Description:Maximal NECA stimulation of adenylate cyclase via adenosine A2 receptor in human platelet membranesMore data for this Ligand-Target Pair
Affinity DataEC50: 178nMAssay Description:In vitro effect on coronary vasodilation in guinea pig heart.More data for this Ligand-Target Pair
Affinity DataEC50: 260nMAssay Description:Potency against human platelet A2 adenosine receptorMore data for this Ligand-Target Pair