Compile Data Set for Download or QSAR
maximum 50k data
Found 32 of ec50 for UniProtKB: P32239
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataEC50:  0.00900nMAssay Description:Ability to stimulate intracellular calcium response was determined using CCK receptor-bearing chinese hamster ovary cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50004477(CCK7 analogue | CHEMBL269016 | N-(1-Carbamoyl-2-ph...)
Affinity DataEC50:  0.100nMAssay Description:Thermodynamic dissociation constant of compound for wild type E. coli dihydrofolate reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50004482(CCK7 analogue | CHEMBL263742 | N-(1-Carbamoyl-2-ph...)
Affinity DataEC50:  0.320nMAssay Description:Thermodynamic dissociation constant of compound for mutant T46A E. coli dihydrofolate reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50004436(3-Acetylamino-N-[1-[1-({[1-{1-[1-(1-carbamoyl-2-ph...)
Affinity DataEC50:  0.5nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50004480(CCK7 analogue | CHEMBL316944)
Affinity DataEC50:  0.640nMAssay Description:Dissociation rate constant of compound for mutant T46A Escherichia coli dihydrofolate reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50421963(CHEMBL2310856)
Affinity DataEC50:  0.700nMAssay Description:Inhibitor constant of compound for wild type E. coli dihydrofolate reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50004437(3-Acetylamino-N-[1-[1-({[1-(1-{[1-(1-carbamoyl-2-p...)
Affinity DataEC50:  0.900nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50004474(CCK7 analogue | CHEMBL316949 | N-(1-Carbamoyl-2-ph...)
Affinity DataEC50:  0.990nMAssay Description:Dissociation rate constant of compound for mutant T46A Escherichia coli dihydrofolate reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50004483(CCK7 analogue | CHEMBL269355)
Affinity DataEC50:  1.30nMAssay Description:Dissociation rate constant of compound for wild type Escherichia coli dihydrofolate reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50004440(3-Acetylamino-N-[1-[1-({[1-{1-[1-(1-carbamoyl-2-ph...)
Affinity DataEC50:  1.40nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataEC50:  2nMAssay Description:Concentration of compound that induced 50% of the maximal contraction in guinea pig gallbladder tissue when tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50004481(CCK7 analogue | CHEMBL99499)
Affinity DataEC50:  2.5nMAssay Description:Dissociation rate constant of compound for mutant T46S Escherichia coli dihydrofolate reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50004439(3-Acetylamino-N-[1-[1-({[1-{1-[1-(1-carbamoyl-2-ph...)
Affinity DataEC50:  3.5nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50004475(CCK7 analogue | CHEMBL439591 | N-(1-Carbamoyl-2-ph...)
Affinity DataEC50:  3.70nMAssay Description:Thermodynamic dissociation constant of compound for mutant T46N E. coli dihydrofolate reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50004489(CCK7 analogue | CHEMBL318010)
Affinity DataEC50:  3.70nMAssay Description:Thermodynamic dissociation constant of compound for wild type E. coli dihydrofolate reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50004438(3-Acetylamino-N-[1-[1-({[1-(1-{1-[(1-carbamoyl-2-p...)
Affinity DataEC50:  4nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50455609(CHEMBL2310857)
Affinity DataEC50:  6.90nMAssay Description:Dissociation rate constant of compound for mutant T46N Escherichia coli dihydrofolate reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50004490(CCK7 analogue | CHEMBL412238 | N-(1-Carbamoyl-2-ph...)
Affinity DataEC50:  15nMAssay Description:Inhibitor constant of compound for mutant T46N E. coli dihydrofolate reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50004435(3-Acetylamino-N-[1-{1-[({[1-{1-[1-(1-carbamoyl-2-p...)
Affinity DataEC50:  26nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50472279(CHEMBL405243)
Affinity DataEC50:  28nMAssay Description:Ability to stimulate intracellular calcium response was determined using CCK receptor-bearing chinese hamster ovary cell lineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50004433(3-Acetylamino-N-[1-[1-({[1-({1-[1-(1-carbamoyl-2-p...)
Affinity DataEC50:  37nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50004488(CCK7 analogue | CHEMBL414793)
Affinity DataEC50:  50nMAssay Description:Dissociation rate constant of compound for mutant T46S Escherichia coli dihydrofolate reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50004492(CCK7 analogue | CHEMBL98720)
Affinity DataEC50:  71nMAssay Description:Dissociation rate constant of compound for wild type Escherichia coli dihydrofolate reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50004434(3-Acetylamino-N-[1-(1-{2-[1-{1-[1-(1-carbamoyl-2-p...)
Affinity DataEC50:  104nMAssay Description:In vitro smooth muscle contraction activity in guinea pig ileum consists of two or three CCK receptor subtypesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50450536(CHEMBL357983)
Affinity DataEC50:  110nMAssay Description:Concentration of compound that induced 50% of the maximal contraction in guinea pig gallbladder tissue when tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50004485(CCK7 analogue | CHEMBL98631)
Affinity DataEC50:  140nMAssay Description:Dissociation rate constant of compound for mutant T46N Escherichia coli dihydrofolate reductaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50472278(CHEMBL410965)
Affinity DataEC50:  150nMAssay Description:Ability to stimulate intracellular calcium response was determined using CCK receptor-bearing chinese hamster ovary cell lineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50450537(CHEMBL146206)
Affinity DataEC50:  210nMAssay Description:Concentration of compound that induced 50% of the maximal contraction in guinea pig gallbladder tissue when tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50472277(CHEMBL438912)
Affinity DataEC50:  280nMAssay Description:Ability to stimulate intracellular calcium response was determined using CCK receptor-bearing chinese hamster ovary cell lineMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50450535(CHEMBL421778)
Affinity DataEC50:  300nMAssay Description:Concentration of compound that induced 50% of the maximal contraction in guinea pig gallbladder tissue when tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50072427(1-(1-(2-(isopropyl(phenyl)amino)-2-oxoethyl)-2,4-d...)
Affinity DataEC50:  1.60E+3nMAssay Description:Concentration of compound that induced 50% of the maximal contraction in guinea pig gallbladder tissue when tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Mayo Clinic And Foundation

Curated by ChEMBL
LigandPNGBDBM50215056(CHEMBL346160)
Affinity DataEC50:  5.60E+3nMAssay Description:Concentration of compound that induced 50% of the maximal contraction in guinea pig gallbladder tissue when tested in vitroMore data for this Ligand-Target Pair
In DepthDetails Article