TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 0.0200nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Compound was evaluated for the binding affinity towards opioid receptor from rat whole brain using [3H]etorpine (33.2 Ci/mmol,0.2nanoM)as radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 0.550nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Compound was evaluated for the binding affinity towards opioid receptor from rat whole brain using [3H]etorpine (33.2 Ci/mmol,0.2nanoM)as radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 3.10nMAssay Description:Compound was evaluated for the binding affinity towards opioid receptor from rat whole brain using [3H]etorpine (33.2 Ci/mmol,0.2nanoM)as radioligandMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 3.30nMAssay Description:Inhibition of human erythrocyte carbonic anhydrase IIMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Compound was evaluated for the inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the presence of NaMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has Muscarinic acetylcholine receptor M2 sub...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 4.30nMAssay Description:Inhibition of human erythrocyte carbonic anhydrase IIMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 6.5nMAssay Description:Inhibition of human erythrocyte carbonic anhydrase IIMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 7.70nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 8.20nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 8.20nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has Muscarinic acetylcholine receptor M2 sub...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 9.10nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:Inhibition of human erythrocyte carbonic anhydrase IIMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 15nMAssay Description:Inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the absence of NaMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has M2 muscarinic receptor subtype.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has M2 muscarinic receptor subtype.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 41nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 49nMAssay Description:In vitro affinity to displace [3H]naloxone from opiate receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 56nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 62nMAssay Description:Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family)More data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: 77nMAssay Description:Compound was evaluated for the inhibition of [3H]- naloxone binding to Opioid receptors in rat brain membrane in the presence of NaMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:In vitro affinity to displace [3H]naloxone from opioid receptor in freshly prepared rat brain homogenatesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rattus norvegicus (rat))
Anaquest Pharmaceuticals
Curated by ChEMBL
Anaquest Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: >100nMAssay Description:Antimuscarinic activity on the acetylcholine-induced inhibition of contraction of guinea pig ileum which has M2 muscarinic receptor subtype.More data for this Ligand-Target Pair