Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of ec50 for monomerid = 50326219
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50326219(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
Affinity DataEC50:  150nMAssay Description:Agonist activity at human muscarinic M1 receptor expressed in CHO-K1 cells assessed as increase of acetylcholine-induced calcium flux by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50326219(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
Affinity DataEC50:  210nMAssay Description:Partial agonist activity at EGFP-fused human full length M1 receptor expressed in HEK293 cells assessed as induction of calcium response by fluoresce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50326219(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
Affinity DataEC50:  450nMAssay Description:Partial agonist activity at EGFP-fused human M1 receptor N-terminal truncated at 17 residues expressed in HEK293 cells assessed as induction of calci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50326219(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
Affinity DataEC50:  720nMAssay Description:Partial agonist activity at EGFP-fused human M1 receptor N-terminal truncated at 11 residues expressed in HEK293 cells assessed as induction of calci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50326219(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
Affinity DataEC50:  740nMAssay Description:Partial agonist activity at human full length M1 receptor expressed in HEK293 cells assessed as induction of calcium response by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed