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Report error Found 6 of ic50 for monomerid = 47032
TargetPhosphoethanolamine/phosphocholine phosphatase(Human)
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM47032(2-[[3-methyl-4-(2,2,2-trifluoroethoxy)-2-pyridinyl...)
Affinity DataIC50:  434nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBMRI, San Diego, C...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetNAD(+) hydrolase SARM1(Human)
Washington University

US Patent
LigandPNGBDBM47032(2-[[3-methyl-4-(2,2,2-trifluoroethoxy)-2-pyridinyl...)
Affinity DataIC50:  3.30E+3nMAssay Description:This assay is an adaptation of the NAD+/NADH Glo assay (Promega G9071). In this assay, NAD+ cycling enzymes convert NAD+ into NADH. In the presence o...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetNAD(+) hydrolase SARM1(Human)
Washington University

US Patent
LigandPNGBDBM47032(2-[[3-methyl-4-(2,2,2-trifluoroethoxy)-2-pyridinyl...)
Affinity DataIC50:  3.50E+3nMAssay Description:Reaction mixtures were prepared on ice by mixing 10 ul of SARM1 SAM-TIR cell lysate (320 fold dilution of lysate 11-3-2016, or 80 fold lysate dilutio...More data for this Ligand-Target Pair
In DepthDetails US Patent

TargetIndoleamine 2,3-dioxygenase 2(Mouse)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM47032(2-[[3-methyl-4-(2,2,2-trifluoroethoxy)-2-pyridinyl...)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of mouse Ido2 transfected in HEK293T cells using L-tryptophan as substrate assessed as kynurenine formation after 45 mins by spectrophotom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Human)
Institute of Clinical Pharmacology

Curated by ChEMBL
LigandPNGBDBM47032(2-[[3-methyl-4-(2,2,2-trifluoroethoxy)-2-pyridinyl...)
Affinity DataIC50:  6.28E+4nMAssay Description:TP_TRANSPORTER: inhibition of Digoxin transepithelial transport (basal to apical) (Digoxin: 5 uM) in Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIndoleamine 2,3-dioxygenase 1(Mouse)
The University of Sydney

Curated by ChEMBL
LigandPNGBDBM47032(2-[[3-methyl-4-(2,2,2-trifluoroethoxy)-2-pyridinyl...)
Affinity DataIC50:  9.40E+4nMAssay Description:Inhibition of mouse Ido1 transfected in HEK293T cells using L-tryptophan as substrate assessed as kynurenine formation after 45 mins by spectrophotom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed