Compile Data Set for Download or QSAR
maximum 50k data
Found 9 of ic50 for monomerid = 50030709
TargetType-2 angiotensin II receptor(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030709(CHEMBL338434 | Pentanoic acid {3-[3-butyl-4-(3-flu...)
Affinity DataIC50:  0.160nMAssay Description:In vitro inhibitory activity against angiotensin II type 2 receptor in rat adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030709(CHEMBL338434 | Pentanoic acid {3-[3-butyl-4-(3-flu...)
Affinity DataIC50:  0.220nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 2 in rat midbrain membrane preparations.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030709(CHEMBL338434 | Pentanoic acid {3-[3-butyl-4-(3-flu...)
Affinity DataIC50:  0.410nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 1 in human adrenal membrane preparations. For this assay, only 0.02%BSA was presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030709(CHEMBL338434 | Pentanoic acid {3-[3-butyl-4-(3-flu...)
Affinity DataIC50:  0.420nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 1 in rabbit aorta membrane preparations.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030709(CHEMBL338434 | Pentanoic acid {3-[3-butyl-4-(3-flu...)
Affinity DataIC50:  0.420nMAssay Description:Antagonist activity at Oryctolagus cuniculus (rabbit) aortic AT1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030709(CHEMBL338434 | Pentanoic acid {3-[3-butyl-4-(3-flu...)
Affinity DataIC50:  0.421nMAssay Description:Antagonist activity at Oryctolagus cuniculus (rabbit) aortic AT1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030709(CHEMBL338434 | Pentanoic acid {3-[3-butyl-4-(3-flu...)
Affinity DataIC50:  0.880nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 2 in human adrenal membrane preparations. For this assay, only 0.02%BSA was presen...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030709(CHEMBL338434 | Pentanoic acid {3-[3-butyl-4-(3-flu...)
Affinity DataIC50:  0.900nMAssay Description:In vitro inhibitory activity against angiotensin II receptor type 1, in human adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-2 angiotensin II receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50030709(CHEMBL338434 | Pentanoic acid {3-[3-butyl-4-(3-flu...)
Affinity DataIC50:  3.80nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor type 2 in human adrenal membrane preparations.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed