Compile Data Set for Download or QSAR
Report error Found 3 of ic50 for monomerid = 50061203
TargetSodium-dependent serotonin transporter(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50061203((R)-3-(4-Ethyl-3-iodo-phenyl)-8-aza-bicyclo[3.2.1]...)
Affinity DataIC50: 0.690nMAssay Description:In vitro inhibitory activity against radioligand [3H]paroxetine binding to serotonin transporter (5-HTT) in rat midbrain tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2012
Entry Details Article
PubMed
TargetTransporter(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50061203((R)-3-(4-Ethyl-3-iodo-phenyl)-8-aza-bicyclo[3.2.1]...)
Affinity DataIC50: 148nMAssay Description:In vitro inhibitory activity against radioligand [3H]-nisoxatine binding to norepinephrine transporter (NET) in rat cortical tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2012
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Research Triangle Institute

Curated by ChEMBL
LigandPNGBDBM50061203((R)-3-(4-Ethyl-3-iodo-phenyl)-8-aza-bicyclo[3.2.1]...)
Affinity DataIC50: 329nMAssay Description:In vitro inhibitory activity against radioligand [3H]-WN 35,428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2012
Entry Details Article
PubMed