Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Antagonist activity at 5-HT2B receptor (unknown origin) expressed in CHO-K1 cells assessed as calcium flux after 60 mins by FLIPR assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 35nMAssay Description:Antagonist activity at 5HT2B (unknown origin) expressed in CHOK1 cells assessed as inhibition of agonist-induced effect preincubated for 60 mins at 3...More data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of human ERG channel by patch clamp assayMore data for this Ligand-Target Pair