Compile Data Set for Download or QSAR
maximum 50k data
Found 6 of ic50 for monomerid = 50395633
TargetEndothelin-1 receptor(Homo sapiens (Human))
Actelion Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50395633(CHEMBL2165332)
Affinity DataIC50:  0.700nMAssay Description:Antagonist activity at ETA receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Actelion Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50395633(CHEMBL2165332)
Affinity DataIC50:  0.700nMAssay Description:Displacement of [I125]ET1 from recombinant ETA receptor expressed in CHO cells after 2 hrs by TopCount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(Homo sapiens (Human))
Actelion Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50395633(CHEMBL2165332)
Affinity DataIC50:  0.700nMAssay Description:Antagonist activity at ETA receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50395633(CHEMBL2165332)
Affinity DataIC50:  441nMAssay Description:Antagonist activity at ETB receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50395633(CHEMBL2165332)
Affinity DataIC50:  441nMAssay Description:Displacement of [I125]ET1 from recombinant ETB receptor expressed in CHO cells after 2 hrs by TopCount analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(Homo sapiens (Human))
Actelion Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50395633(CHEMBL2165332)
Affinity DataIC50:  441nMAssay Description:Antagonist activity at ETB receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed