Compile Data Set for Download or QSAR
maximum 50k data
Found 7 of ic50 for monomerid = 50428067
TargetPlasminogen(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50428067(CL-65336 | Cyklokapron | Lysteda | TRANEXAMIC ACID...)
Affinity DataIC50:  3.10E+3nMAssay Description:Binding affinity to full length Glu-plasminogen in human plasma assessed as inhibition of interaction with fibrin in presence of tPAMore data for this Ligand-Target Pair
TargetPlasminogen(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50428067(CL-65336 | Cyklokapron | Lysteda | TRANEXAMIC ACID...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of plasminogen/fibrinogen interaction in pooled citrated human platelet-poor plasma assessed as inhibition of lysis of CaCl2/t-PA-induced ...More data for this Ligand-Target Pair
TargetPlasminogen(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50428067(CL-65336 | Cyklokapron | Lysteda | TRANEXAMIC ACID...)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of human Glu-plasminogen/fibrinogen interaction in HEPES buffer assessed as inhibition of lysis of thrombin-induced clot preincubated for ...More data for this Ligand-Target Pair
TargetPlasminogen(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50428067(CL-65336 | Cyklokapron | Lysteda | TRANEXAMIC ACID...)
Affinity DataIC50:  1.20E+4nMAssay Description:Binding affinity to human full length Glu-plasminogen in buffer assessed as inhibition of interaction with fibrin preincubated for 15 mins followed b...More data for this Ligand-Target Pair
TargetPlasminogen(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50428067(CL-65336 | Cyklokapron | Lysteda | TRANEXAMIC ACID...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of human plasmin assessed as inhibition of fibrinolysis in presence of fibrinogenMore data for this Ligand-Target Pair
TargetPlasminogen(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50428067(CL-65336 | Cyklokapron | Lysteda | TRANEXAMIC ACID...)
Affinity DataIC50:  2.00E+6nMAssay Description:Inhibition of plasmin (unknown origin) after 18 hrs by arianor mahogany dye-based fibrin plate assayMore data for this Ligand-Target Pair
TargetPlasminogen(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50428067(CL-65336 | Cyklokapron | Lysteda | TRANEXAMIC ACID...)
Affinity DataIC50:  1.00E+7nMAssay Description:Inhibition of human plasmin assessed as inhibition of fibrinogenolysis in presence of fibrinogenMore data for this Ligand-Target Pair