Report error Found 26 of ic50 for monomerid = 90787
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
Budapest University of Technology and Economics
Curated by ChEMBL
Budapest University of Technology and Economics
Curated by ChEMBL
Affinity DataIC50: 1.68E+3nMAssay Description:H-bonding interaction between amino acid residue (Asn-137) of Sodium- and chloride-dependent GABA transporter 1TM3 and compoundMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
Budapest University of Technology and Economics
Curated by ChEMBL
Budapest University of Technology and Economics
Curated by ChEMBL
Affinity DataIC50: 1.68E+3nMAssay Description:H-bonding interaction between amino acid residue (Asn-137) of Sodium- and chloride-dependent GABA transporter 1TM3 and compoundMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
Budapest University of Technology and Economics
Curated by ChEMBL
Budapest University of Technology and Economics
Curated by ChEMBL
Affinity DataIC50: 1.68E+3nMAssay Description:H-bonding interaction between amino acid residue (Asn-137) of Sodium- and chloride-dependent GABA transporter 1TM3 and compoundMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
Budapest University of Technology and Economics
Curated by ChEMBL
Budapest University of Technology and Economics
Curated by ChEMBL
Affinity DataIC50: 2.59E+3nMAssay Description:H-bonding interaction between amino acid residue (Tyr-140) of Sodium- and chloride-dependent GABA transporter 1TM3 and compound was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
Budapest University of Technology and Economics
Curated by ChEMBL
Budapest University of Technology and Economics
Curated by ChEMBL
Affinity DataIC50: 2.59E+3nMAssay Description:H-bonding interaction between amino acid residue (Tyr-140) of Sodium- and chloride-dependent GABA transporter 1TM3 and compound was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
Budapest University of Technology and Economics
Curated by ChEMBL
Budapest University of Technology and Economics
Curated by ChEMBL
Affinity DataIC50: 2.65E+3nMAssay Description:H-bonding interaction between amino acid residue (Tyr-140) of Sodium- and chloride-dependent GABA transporter 1TM3 and compound was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
Budapest University of Technology and Economics
Curated by ChEMBL
Budapest University of Technology and Economics
Curated by ChEMBL
Affinity DataIC50: 2.65E+3nMAssay Description:H-bonding interaction between amino acid residue (Tyr-140) of Sodium- and chloride-dependent GABA transporter 1TM3 and compound was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
Budapest University of Technology and Economics
Curated by ChEMBL
Budapest University of Technology and Economics
Curated by ChEMBL
Affinity DataIC50: 2.66E+3nMAssay Description:H-bonding interaction between amino acid residue (Thr-89) of Sodium- and chloride-dependent GABA transporter 1TM2 and compoundMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
Budapest University of Technology and Economics
Curated by ChEMBL
Budapest University of Technology and Economics
Curated by ChEMBL
Affinity DataIC50: 2.66E+3nMAssay Description:H-bonding interaction between amino acid residue (Thr-89) of Sodium- and chloride-dependent GABA transporter 1TM2 and compoundMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
Budapest University of Technology and Economics
Curated by ChEMBL
Budapest University of Technology and Economics
Curated by ChEMBL
Affinity DataIC50: 2.77E+3nMAssay Description:H-bonding interaction between amino acid residue (Ser-133) of Sodium- and chloride-dependent GABA transporter 1TM3 and compound was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
Budapest University of Technology and Economics
Curated by ChEMBL
Budapest University of Technology and Economics
Curated by ChEMBL
Affinity DataIC50: 2.77E+3nMAssay Description:H-bonding interaction between amino acid residue (Ser-133) of Sodium- and chloride-dependent GABA transporter 1TM3 and compound was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
Budapest University of Technology and Economics
Curated by ChEMBL
Budapest University of Technology and Economics
Curated by ChEMBL
Affinity DataIC50: 2.79E+3nMAssay Description:H-bonding interaction between amino acid residue (Asn-137) of Sodium- and chloride-dependent GABA transporter 1TM3 and compoundMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
Budapest University of Technology and Economics
Curated by ChEMBL
Budapest University of Technology and Economics
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:H-bonding interaction between amino acid residue (Ser-133) of Sodium- and chloride-dependent GABA transporter 1TM3 and compound was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
Budapest University of Technology and Economics
Curated by ChEMBL
Budapest University of Technology and Economics
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:H-bonding interaction between amino acid residue (Ser-133) of Sodium- and chloride-dependent GABA transporter 1TM3 and compound was determinedMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Mouse)
Ludwig Maximilians University At Munich
Curated by ChEMBL
Ludwig Maximilians University At Munich
Curated by ChEMBL
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of [3H]GABA uptake at mouse GAT1 expressed in HEK293 cells after 25 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Human)
Synaptic Pharmaceutical
Curated by ChEMBL
Synaptic Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibitory activity against human GABA transporter-1 (hGAT1)More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Human)
Synaptic Pharmaceutical
Curated by ChEMBL
Synaptic Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of human GAT1 expressed in COS cells assessed as decrease in [3H]GABA uptake after 10 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 1(Rat)
Budapest University of Technology and Economics
Curated by ChEMBL
Budapest University of Technology and Economics
Curated by ChEMBL
Affinity DataIC50: 2.09E+4nMAssay Description:Inhibition of mouse GAT1 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 2(Rat)
Synaptic Pharmaceutical
Curated by ChEMBL
Synaptic Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 5.80E+4nMAssay Description:Inhibitory activity against rat GABA transporter-2 (rGAT2)More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 2(Human)
Zentrum F£R Pharmaforschung
Curated by ChEMBL
Zentrum F£R Pharmaforschung
Curated by ChEMBL
Affinity DataIC50: 6.60E+4nMAssay Description:Binding affinity to GAT2More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 2(Mouse)
University of Louvain
Curated by ChEMBL
University of Louvain
Curated by ChEMBL
Affinity DataIC50: 7.24E+4nMAssay Description:Inhibition of mouse GAT2 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 3(Human)
Zentrum F£R Pharmaforschung
Curated by ChEMBL
Zentrum F£R Pharmaforschung
Curated by ChEMBL
Affinity DataIC50: 1.10E+5nMAssay Description:Binding affinity to GAT3More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 3(Mouse)
University of Louvain
Curated by ChEMBL
University of Louvain
Curated by ChEMBL
Affinity DataIC50: 1.15E+5nMAssay Description:Inhibition of mouse GAT3 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent GABA transporter 3(Human)
Zentrum F£R Pharmaforschung
Curated by ChEMBL
Zentrum F£R Pharmaforschung
Curated by ChEMBL
Affinity DataIC50: 1.19E+5nMAssay Description:Inhibitory activity against human sodium and chloride dependent GABA transporter 3More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Mouse)
University of Louvain
Curated by ChEMBL
University of Louvain
Curated by ChEMBL
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of mouse BGT1 mediated [3]GABA uptake expressed in HEK293 cells after 3 mins by scintillation countingMore data for this Ligand-Target Pair
TargetSodium- and chloride-dependent betaine transporter(Human)
Synaptic Pharmaceutical
Curated by ChEMBL
Synaptic Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 1.87E+6nMAssay Description:Inhibition of human GABA transporter (hBGT-1) activity.More data for this Ligand-Target Pair
