Affinity DataKd: 1.20nMAssay Description:Binding affinity to recombinant human HSP90 alpha by Surface plasmon resonance analysisMore data for this Ligand-Target Pair
Affinity DataKd: 1.80nMAssay Description:Binding affinity to recombinant human HSP90alpha by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Affinity DataKd: 2.20nMAssay Description:Binding affinity to human Hsp90 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha/90-beta(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKd: 19nMAssay Description:Binding affinity to HSP90 (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-alpha [1-236](Homo sapiens (Human))
University Of Texas Southwestern Medical Center
University Of Texas Southwestern Medical Center
Affinity DataKd: 46.3nMpH: 7.5 T: 2°CAssay Description:The PDK2 or Hsp90 N-terminal domain protein was dialyzed against 1 liter of thedialysis buffer containing 50 mM Tris-Cl, pH 7.5, 50 mM KCl, 1 mM MgCl...More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
University Of Texas Southwestern Medical Center
University Of Texas Southwestern Medical Center
Affinity DataKd: 1.86E+4nMpH: 7.5 T: 2°CAssay Description:The PDK2 or Hsp90 N-terminal domain protein was dialyzed against 1 liter of thedialysis buffer containing 50 mM Tris-Cl, pH 7.5, 50 mM KCl, 1 mM MgCl...More data for this Ligand-Target Pair
TargetVirulence sensor histidine kinase PhoQ(Salmonella typhimurium (strain LT2 / SGSC1412 / AT...)
Williams College
Curated by ChEMBL
Williams College
Curated by ChEMBL
Affinity DataKd: 7.15E+5nMAssay Description:Binding affinity to recombinant Salmonella typhimurium 15N-labeled PhoQ catalytic domain (332 to 487 residues) expressed in Escherichia coli XA90 ass...More data for this Ligand-Target Pair