Compile Data Set for Download or QSAR
Report error Found 6 of ki for monomerid = 13936
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13936BDBM13936(N-1465 | Ace-T-I-Nle-r-Nle-Q-R | Ac-Thr-Ile-Nle-r-...)
Affinity DataKi:  776nMAssay Description:Binding affinity to HIV-1 proteaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2014
Entry Details Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 13936BDBM13936(N-1465 | Ace-T-I-Nle-r-Nle-Q-R | Ac-Thr-Ile-Nle-r-...)
Affinity DataKi:  780nMAssay Description:Binding affinity against HIV-1 aspartic proteinase was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2012
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599,Q508K,L534I,L564I,C568A,C596A,L525I](Human immunodeficiency virus type 1)
Georgia State University

LigandChemical structure of BindingDB Monomer ID 13936BDBM13936(N-1465 | Ace-T-I-Nle-r-Nle-Q-R | Ac-Thr-Ile-Nle-r-...)
Affinity DataKi:  2.00E+3nM ΔG°:  -32.2kJ/molepH: 5.0 T: 2°CAssay Description:The Ki values were obtained from the IC50 values estimated from an inhibitor dose-response curve with the spectroscopic assay and the chromogenic sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2007
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599,Q508K,L534I,L564I,C568A,C596A](Human immunodeficiency virus type 1)
Georgia State University

LigandChemical structure of BindingDB Monomer ID 13936BDBM13936(N-1465 | Ace-T-I-Nle-r-Nle-Q-R | Ac-Thr-Ile-Nle-r-...)
Affinity DataKi:  2.17E+3nM ΔG°:  -32.0kJ/molepH: 5.0 T: 2°CAssay Description:The Ki values were obtained from the IC50 values estimated from an inhibitor dose-response curve with the spectroscopic assay and the chromogenic sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2007
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599,Q508K,L534I,L564I,C568A,C596A,G574S](Human immunodeficiency virus type 1)
Georgia State University

LigandChemical structure of BindingDB Monomer ID 13936BDBM13936(N-1465 | Ace-T-I-Nle-r-Nle-Q-R | Ac-Thr-Ile-Nle-r-...)
Affinity DataKi:  3.30E+3nM ΔG°:  -31.0kJ/molepH: 5.0 T: 2°CAssay Description:The Ki values were obtained from the IC50 values estimated from an inhibitor dose-response curve with the spectroscopic assay and the chromogenic sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2007
Entry Details Article
PubMed
TargetDimer of Gag-Pol polyprotein [501-599,Q508K,L534I,L564I,C568A,C596A,I551V](Human immunodeficiency virus type 1)
Georgia State University

LigandChemical structure of BindingDB Monomer ID 13936BDBM13936(N-1465 | Ace-T-I-Nle-r-Nle-Q-R | Ac-Thr-Ile-Nle-r-...)
Affinity DataKi:  4.10E+4nM ΔG°:  -24.8kJ/molepH: 5.0 T: 2°CAssay Description:The Ki values were obtained from the IC50 values estimated from an inhibitor dose-response curve with the spectroscopic assay and the chromogenic sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/19/2007
Entry Details Article
PubMed