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Report error Found 2 of ki for monomerid = 24182

Gamma-aminobutyric acid (GABA) B receptor 1/type B receptor subunit 2 [41-940](Rat)
Astrazeneca

BDBM24182(4-amino-3-(4-chlorophenyl)butanoic acid | Baclofen...)

Ki: 220nM ΔG°: -37.6kJ/mole EC50: 750nMpH: 7.4 T: 22°CAssay Description:Inhibition of [3H]GABA binding at GABAB receptor sites in rat brain synaptic membranes by test compounds was measured using a filtration binding assa...More data for this Ligand-Target Pair

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3D Structure (crystal)

Gamma-aminobutyric acid type B receptor subunit 1/2(Human)
Purdue University

Curated by ChEMBL

BDBM24182(4-amino-3-(4-chlorophenyl)butanoic acid | Baclofen...)

Ki: 6.00E+3nMAssay Description:Displacement of [3H]CGP54626 from GABA-B receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
B.MOAD DrugBank antibodypedia GoogleScholar

Purchase ChEBI
CHEMBL DrugBank MCE
PC cid PC sid PDB Patents Similars

Details Article PubMed DrugBank
PDB

3D Structure (crystal)