Report error Found 68 of ki for monomerid = 50085658
Affinity DataKi: 0.210nMAssay Description:Displacement of [3H]N6-R-phenylisopropyladenosine from mouse A1A adenosine receptor expressed in CHO cell membranes after 60 mins by scintillation pr...More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in pig cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.340nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in bovine cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.350nMAssay Description:Inhibitory activity at Adenosine A1 receptor by inhibition of [3H]CHA binding to bovine brain cortical membranes.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rat)
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
TargetAdenosine receptor A1(Rat)
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 0.600nMAssay Description:Tested for the binding affinity of A1 receptor by displacing the [3H]-PIA in rat brain membranesMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rat)
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 0.600nMAssay Description:Binding affinity for Adenosine A1 receptor using [3H]- CHA or [3H]- PIAMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rat)
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 0.600nMAssay Description:Inhibition of [3H]- (R)-P1A binding to adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]CCPA from human recombinant adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Displacement of [3H]CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Displacement of [3H]N6-R-phenylisopropyladenosine from human A1A adenosine receptor expressed in CHO cell membranes after 60 mins by scintillation pr...More data for this Ligand-Target Pair
Affinity DataKi: 0.830nMAssay Description:Displacement of [3H]R-PIA or [3H]CGS 21680 from human adenosine A1 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.830nM ΔG°: -48.2kJ/molepH: 7.4 T: 2°CAssay Description:Membranes for radioligand binding experiments are prepared from fresh or frozen cells as described in Klotz et al., Naunyn-Schmiedeberg's Arch. Pharm...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Ex vivo inhibition of guinea pig ileum twitch via Adenosine A1 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-CCPA from human A1 receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rat)
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor of rat brainMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rat)
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 1.30nMAssay Description:Affinity for adenosine A1 receptor assayed in a competition assay in rat brain using [3H]-CHA as radioligandMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rat)
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 1.30nMAssay Description:Binding affinity against adenosine A1 receptor from rat brain using [3H]CHA as a radioligand.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rat)
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]R-PIA from rat brain membrane Adenosine A1 receptorMore data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rat)
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 1.5nMAssay Description:Tested for inhibition of adenosine A1 receptor binding to rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:In vitro binding affinity towards human adenosine A1 receptor by [3H]DPCPX displacement.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rat)
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 7.43nMAssay Description:Binding affinity for adenosine A1 receptor was assayed by displacement of [3H]DPCPX from rat cortical membranes.More data for this Ligand-Target Pair
TargetAdenosine receptor A1(Rat)
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
National Institutes of Diabetes and Digestive and Kidney Diseases
Curated by PDSP Ki Database
Affinity DataKi: 9.47nMAssay Description:Affinity towards adenosine A1 receptor from rat cortical membranes using [3H]DPCPXMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 15.1nMAssay Description:Binding affinity to human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 15.3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 90 minsMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [125I]N6-(4-amino-3-iodobenzyl)adenosine-5-N-methyluronamide from mouse A3A adenosine receptor expressed in CHO cell membranes after ...More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:In vitro inhibition of human neutrophil activation via Adenosine A2A receptor.More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [3H]-HEMADO from human A3 receptor stably expressed in CHO cell membranes by radioligand competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Inhibitory activity against Adenosine A3 receptor by inhibiting specific [3H](R)-PIA binding to rat testis membranesMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Binding affinity in membrane of CHO cell stably expressing recombinant human Adenosine A3 receptor in the presence of GTPgammaS using [3H]8-ethyl-4-m...More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Displacement of [125I]N6-(4-amino-3-iodobenzyl)adenosine-5-N-methyluronamide from human A3A adenosine receptor expressed in CHO cell membranes after ...More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Binding affinity to human adenosine A3 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Binding affinity to Adenosine receptor A3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Affinity for human Adenosine A3 receptor expressed in CHO cellMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Bnding affinity in membrane of CHO cell stably expressing recombinant human Adenosine A3 receptor using [3H]8-ethyl-4-methyl-2-phenyl-(8R)-4,5,7,8-te...More data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Agonist activity at human recombinant adenosine A2B receptor expressed in CHO cells assessed as activation of adenylyl cyclase activityMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity towards Adenosine A3 receptor (W243 mutant receptor)More data for this Ligand-Target Pair
Affinity DataKi: 114nMAssay Description:Binding affinity towards human Adenosine A3 receptor wild typeMore data for this Ligand-Target Pair
Affinity DataKi: 204nMAssay Description:Affinity towards Adenosine A3 receptor expressed in HEK 293 cells using [125I]AB-MECA radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 237nMAssay Description:Displacement of [125I]- AB-MECA from rat adenosine A3 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 237nMAssay Description:Binding affinity to rat adenosine A3 receptor in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 237nMAssay Description:Tested for the binding affinity of A3 receptor by displacing N6-[[125I]-4-amino-3-iodobenzyl]-adenosine-5''-N-methyluronamide from membranes of CHO c...More data for this Ligand-Target Pair
Affinity DataKi: 281nMAssay Description:Inhibition of [125 I]-IABMECA binding to human adenosine A3 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 580nMAssay Description:Inhibitory activity at Adenosine A2A receptor by inhibition of [3H]-CGS- 21680 binding to bovine striatal membranes.More data for this Ligand-Target Pair
Affinity DataKi: 605nMAssay Description:Displacement of specific [3H]-CGS- 21680 binding to adenosine A2A receptor in rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 639nMAssay Description:Tested for binding affinity towards human adenosine A2A receptor using [3H]ZM-241385 as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 640nMAssay Description:Binding affinity for adenosine A2A receptor was determined by displacement of [3H]-DPCPX from rat striatal membranes.More data for this Ligand-Target Pair
Affinity DataKi: 650nMAssay Description:Binding affinity against adenosine A2a receptor from rat striatum using [3H]-CGS- 21680 as a radioligand.More data for this Ligand-Target Pair
