Compile Data Set for Download or QSAR
maximum 50k data
Found 2 of ki for monomerid = 50100422
TargetAdenosine receptor A3(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50100422((1R,2S,4S,5S)-4-(6-Cyclopentylamino-purin-9-yl)-1-...)
Affinity DataKi:  2.88E+3nMAssay Description:Ability to displace specific radioligand [125I]AB-MECA binding at human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50100422((1R,2S,4S,5S)-4-(6-Cyclopentylamino-purin-9-yl)-1-...)
Affinity DataKi:  5.11E+3nMAssay Description:Ability to displace specific radioligand [3H]R-PIA binding at Adenosine A1 receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed