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Found 4 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 1A' and Ligand = 'BDBM50051164'
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50051164(2-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-butyl]-isoi...)
Affinity DataKi:  140nMAssay Description:Binding affinity towards 5-hydroxytryptamine 1A receptor in the rat brain (hippocampus) using [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Polish Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50051164(2-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-butyl]-isoi...)
Affinity DataKi:  355nMAssay Description:Ability of the compound to displace [3H]-8-OH-DPAT from 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50051164(2-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-butyl]-isoi...)
Affinity DataKi:  499nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in cell membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Florida A&M University

Curated by ChEMBL
LigandPNGBDBM50051164(2-[4-(3,4-Dihydro-1H-isoquinolin-2-yl)-butyl]-isoi...)
Affinity DataKi:  501nMAssay Description:Displacement of [3H]8-OH-DPAT from human 5-HT1A receptor expressed in cell membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed