Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 3A' and Ligand = 'BDBM50000492'
Target5-hydroxytryptamine receptor 3A(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50000492BDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  0.320nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/2/2012
Entry Details
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
University of Missouri

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000492BDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  0.390nMAssay Description:Displacement of [3H]GR65630 from 5-HT3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Human)
University of Missouri

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000492BDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  0.398nMAssay Description:Displacement of [3H]GR65630 from 5-HT3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50000492BDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKd:  0.600nMAssay Description:Compound was tested for its antagonistic activity against 5-hydroxytryptamine 3 receptor in rat brain using [3H]zacopride as the radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 3A(Human)
University of Missouri

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000492BDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  0.700nMAssay Description:In vitro binding affinity for the 5-hydroxytryptamine 3 receptor was determined with NG-108-15 mouse neuroblastoma-glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2012
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 3A(Guinea pig)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50000492BDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  0.950nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/2/2012
Entry Details
PubMed
Target5-hydroxytryptamine receptor 3A(Rat)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50000492BDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  3.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/2/2012
Entry Details
PubMed
Target5-hydroxytryptamine receptor 3A(Guinea pig)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50000492BDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi:  5.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/2/2012
Entry Details
PubMed
Target5-hydroxytryptamine receptor 3A(Guinea pig)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50000492BDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/2/2012
Entry Details
PubMed
Target5-hydroxytryptamine receptor 3A(Guinea pig)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50000492BDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/2/2012
Entry Details
PubMed
Target5-hydroxytryptamine receptor 3A(Guinea pig)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50000492BDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/2/2012
Entry Details
PubMed
Target5-hydroxytryptamine receptor 3A(Guinea pig)
Syntex Discovery Research

Curated by PDSP Ki Database
LigandChemical structure of BindingDB Monomer ID 50000492BDBM50000492(ZACOPRIDE,R | 4-Amino-N-(1-aza-bicyclo[2.2.2]oct-3...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/2/2012
Entry Details
PubMed