Found 6 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 4' and Ligand = 'BDBM50327858'
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
University Of Oslo
Curated by PDSP Ki Database
University Of Oslo
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
University Of Oslo
Curated by PDSP Ki Database
University Of Oslo
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
National Institute Of Mental Health
Curated by ChEMBL
National Institute Of Mental Health
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]GR113808 from 5HT4 receptor in guinea pig striatal membranesMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
University Of Oslo
Curated by PDSP Ki Database
University Of Oslo
Curated by PDSP Ki Database
Affinity DataKi: 2.20nMAssay Description:Displacement of [3H]GR113808 from human recombinant 5HT4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKd: 0.0800nMAssay Description:Binding affinity to 5HT4 receptor in pig striatal membranesMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
University Of Oslo
Curated by PDSP Ki Database
University Of Oslo
Curated by PDSP Ki Database
Affinity DataEC50: 13nMAssay Description:Agonist activity at 5HT4 receptor expressed in HEK293/L9 cells by cAMP assayMore data for this Ligand-Target Pair