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Found 2 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 6' and Ligand = 'BDBM50562747'
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50562747(CHEMBL4756814)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-LSD from human 5HT6R expressed in HEK293 cell membranes incubated for 1 hr by micro-beta plate reader based analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Palack£

Curated by ChEMBL
LigandPNGBDBM50562747(CHEMBL4756814)
Affinity DataIC50:  5.40nMAssay Description:Neutral antagonist activity at 5HT6R (unknown origin) expressed in 1321N1 cells co-expressing CAMYEL assessed as inhibition of WAY181187-induced cAMP...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed