Affinity DataKi: 13nMAssay Description:Inhibition of adenylate cyclase via adenosine A1 receptors in rat fat cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Binding affinity against low affinity component of adenosine A1 receptors from rat brain membranes using [3H]-DPCPXMore data for this Ligand-Target Pair
Affinity DataKi: 98nMAssay Description:Displacement of [3H]CHA from Adenosine A1 receptor of rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 103nMAssay Description:Binding affinity against adenosine A1 receptor from rat brain membranes using [3H]cyclohexyladenosine as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Inhibition of [3H]CHA binding to adenosine A1 receptor from rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Binding affinity against adenosine A1 receptor in rat brain membranes using [3H]CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 147nMAssay Description:Binding affinity against adenosine A1 receptor using [3H]-CHA or [3H]PIA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 633nMAssay Description:Binding affinity against low affinity component of adenosine A1 receptors from rat brain membranes using [3H]-DPCPXMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Binding affinity against high affinity component of adenosine A1 receptors from rat brain membranes using [3H]DPCPXMore data for this Ligand-Target Pair
Affinity DataEC50: >1nMAssay Description:Adenosine A1 receptor mediated negative chronotropic activity in spontaneously beating rat atriaMore data for this Ligand-Target Pair