Report error Found 36 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50207816'
Affinity DataKi: 0.300nMAssay Description:Affinity for Adenosine A1 receptor using [N6-[(3-[125I]-iodo-4-aminophenyl)ethyl]adenosine in calf brainMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Affinity for adenosine A1 receptor using [3H]N6-(phenylisopropyl)adenosine (R)-[3H]-PIA as a radioligand in rat brain.More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]DPCPX binding to adenosine A1 receptor of rat brain cortical membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of (R)-N6-([3H]-phenylisopropyl) adenosine binding to adenosine A1 receptor from rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity towards adenosine A1 receptor in rat cortical membranes using N6-[3H]cyclohexyladenosine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of binding of 1 nM [3H]N-6-(phenylisopropyl)adenosine to adenosine A1 receptor in rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity for adenosine A1 receptor using [3H]- CHA or [3H]- PIAMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Antagonist activity against adenosine A1 receptor in rat brain membrane in presence of [3H]-R-PIA radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-PIA from adenosine A1 receptors of rat brain membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of [3H]- PIA binding at adenosine A1 receptor on rat cerebral cortex membranes.More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Binding affinity towards adenosine A1 receptor in rat cerebral cortical membranes by [3H]-cyclohexyladenosine displacement.More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity towards rat Adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity at bovine Adenosine A1 receptor.More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Ability to displace the specific binding of [3H]CHA to adenosine A1 receptor from bovine brain cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 6.82nMAssay Description:Antagonist activity against recombinant human adenosine A1 receptor expressed in HEK-293 cells in presence of [125I]-IABA radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 8.30nMAssay Description:Antagonist activity at human adenosine A1 receptor assessed as cAMP level by cell based assayMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in HEK293T cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in HEK293T cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity against adenosine A1 receptor from guinea pig forebrain membranes, using N6-[3H]-cyclohexyladenosine as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Binding affinity against adenosine A1 receptor in guinea pig forebrain membranes using N6-[3H]cyclohexyladenosine as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Displacement of [3H]DPCPX from human A1AR expressed in CHO cell membrane incubated for 60 mins by microbeta trilux scintillation counter analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.91E+4nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in human CHO cells incubated for 30 mins by fluorescence polarization binding as...More data for this Ligand-Target Pair
Affinity DataKd: 0.170nMAssay Description:Antagonist activity against beta-1 adrenergic receptor in isolated guinea pig atriaMore data for this Ligand-Target Pair
