Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50232154'
TargetAdenosine receptor A1(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232154BDBM50232154(N-(2-furan-2-yl-6-pyrazol-1-yl-pyrimidin-4-yl)-ace...)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]DPCPX form human adenosine A1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232154BDBM50232154(N-(2-furan-2-yl-6-pyrazol-1-yl-pyrimidin-4-yl)-ace...)
Affinity DataKi:  9.20nMAssay Description:Binding affinity at adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232154BDBM50232154(N-(2-furan-2-yl-6-pyrazol-1-yl-pyrimidin-4-yl)-ace...)
Affinity DataKi:  9.20nMAssay Description:Displacement of [3H]DPCPX from human recombinant adenosine A1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetAdenosine receptor A1(Human)
Neurocrine Biosciences

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50232154BDBM50232154(N-(2-furan-2-yl-6-pyrazol-1-yl-pyrimidin-4-yl)-ace...)
Affinity DataKi:  10nMAssay Description:Inhibition of human recombinant adenosine A1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed