Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A1' and Ligand = 'BDBM50597192'
TargetAdenosine receptor A1(Human)
University of Cambridge

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50597192BDBM50597192(CHEMBL5175347)
Affinity DataEC50:  0.977nMAssay Description:Antagonist activity at human wild type A1R expressed in CHO-K1 cells assessed as inhibition of forskolin/ NECA-stimulated cAMP accumulation by measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetAdenosine receptor A1(Human)
University of Cambridge

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50597192BDBM50597192(CHEMBL5175347)
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of CA200645 from NLuc human A1 receptor expressed in HEK293 cells assessed as inhibition constant by NanoBRET binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed