Affinity DataKi: 1.10nMAssay Description:Binding of Adenosine A2 receptor in whole rat brain membrane using [3H]CHA as a RadioligandMore data for this Ligand-Target Pair
Affinity DataKi: 321nMAssay Description:Tested for inhibition of adenosine A2 receptor binding to rat brainMore data for this Ligand-Target Pair
Affinity DataKi: 336nMAssay Description:Binding affinity against adenosine A2 receptor from rat striatum using [3H]NECA as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 421nMAssay Description:Binding affinity against adenosine A2 receptor in rat striatal membranes using [3H]NECA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 460nMAssay Description:Binding affinity towards adenosine A2 receptor on rat striatal membrane using [3H]NECA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 460nMAssay Description:Binding affinity at adenosine A2 receptor from rat striatal membranes by [3H]NECA displacement.More data for this Ligand-Target Pair
Affinity DataKi: 462nMAssay Description:Affinity for Adenosine A2 receptor determined by [3H]NECA binding to rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataKi: 462nMAssay Description:Binding affinity against Adenosine A2 receptor using [3H]NECA with 50 nM CPA in rat striatal brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 462nMAssay Description:Displacement of [3H]-NECA from adenosine A2 receptor of rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 510nMAssay Description:Inhibition of [3H]- NECA binding to adenosine receptor A2More data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Binding affinity against adenosine A1 receptors from rat brain membranes using [3H]CCPAMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Inhibition of Adenylate cyclase activity in rat fat cell membrane at adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.40E+3nMAssay Description:Binding affinity against high affinity component of adenosine A1 receptors from rat brain membranes using [3H]DPCPXMore data for this Ligand-Target Pair
Affinity DataIC50: 1.16E+3nMAssay Description:Concentration required for 50% inhibition of [3H]NECA binding on rat brain adenosine A2 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 2.20E+3nMAssay Description:Stimulation of adenylate cyclase activity in human platelet membrane at A2 receptorMore data for this Ligand-Target Pair