Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50109461'
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50109461(CHEMBL324735 | MRE 3046F20 | 1-(2-Furan-2-yl-8-met...)
Affinity DataKi:  0.160nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50109461(CHEMBL324735 | MRE 3046F20 | 1-(2-Furan-2-yl-8-met...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]MRE3008-F20 from human A3 receptors expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50109461(CHEMBL324735 | MRE 3046F20 | 1-(2-Furan-2-yl-8-met...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]-MRE 3008-F20 from Human Adenosine A3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50109461(CHEMBL324735 | MRE 3046F20 | 1-(2-Furan-2-yl-8-met...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2016
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50109461(CHEMBL324735 | MRE 3046F20 | 1-(2-Furan-2-yl-8-met...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]MRE 3008F20 from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50109461(CHEMBL324735 | MRE 3046F20 | 1-(2-Furan-2-yl-8-met...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]MRE3008-F20 from human A3 receptor expressed in CHO cells by scintillation counterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2017
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50109461(CHEMBL324735 | MRE 3046F20 | 1-(2-Furan-2-yl-8-met...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]MRE3008-F20 from human Adenosine A3 receptor expressed in HEK cells; range 0.13-0.20More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50109461(CHEMBL324735 | MRE 3046F20 | 1-(2-Furan-2-yl-8-met...)
Affinity DataKi:  0.160nMAssay Description:Binding affinity for human adenosine A3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50109461(CHEMBL324735 | MRE 3046F20 | 1-(2-Furan-2-yl-8-met...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]-MRE3008F20 from human recombinant adenosine A3 receptor expressed in HEK293 cells after 120 mins by scintillation counting analy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2016
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50109461(CHEMBL324735 | MRE 3046F20 | 1-(2-Furan-2-yl-8-met...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50109461(CHEMBL324735 | MRE 3046F20 | 1-(2-Furan-2-yl-8-met...)
Affinity DataKi:  1.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50109461(CHEMBL324735 | MRE 3046F20 | 1-(2-Furan-2-yl-8-met...)
Affinity DataKi:  1.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50109461(CHEMBL324735 | MRE 3046F20 | 1-(2-Furan-2-yl-8-met...)
Affinity DataIC50: 2nMAssay Description:Inhibition of IB-MECA agonist-mediated cAMP production in membranes of CHO cells expressing human Adenosine A3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50109461(CHEMBL324735 | MRE 3046F20 | 1-(2-Furan-2-yl-8-met...)
Affinity DataIC50: 2.10nMAssay Description:Inhibitory activity against Human Adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
National University of Singapore

Curated by ChEMBL
LigandPNGBDBM50109461(CHEMBL324735 | MRE 3046F20 | 1-(2-Furan-2-yl-8-met...)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed