Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50109477'
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50109477(1-(4-bromophenyl)-3-(2-(furan-2-yl)-8-methyl-8H-py...)
Affinity DataKi:  0.460nMAssay Description:Binding affinity for human adenosine A3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50109477(1-(4-bromophenyl)-3-(2-(furan-2-yl)-8-methyl-8H-py...)
Affinity DataKi:  0.460nMAssay Description:Displacement of [3H]MRE3008-F20 from human Adenosine A3 receptor expressed in HEK cells; range 0.39-0.54More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50109477(1-(4-bromophenyl)-3-(2-(furan-2-yl)-8-methyl-8H-py...)
Affinity DataKi:  0.460nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50109477(1-(4-bromophenyl)-3-(2-(furan-2-yl)-8-methyl-8H-py...)
Affinity DataKi:  0.460nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50109477(1-(4-bromophenyl)-3-(2-(furan-2-yl)-8-methyl-8H-py...)
Affinity DataKi:  0.460nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2020
Entry Details Article

TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50109477(1-(4-bromophenyl)-3-(2-(furan-2-yl)-8-methyl-8H-py...)
Affinity DataIC50: 4.20nMAssay Description:Inhibition of IB-MECA agonist-mediated cAMP production in CHO cell membranes expressing human Adenosine A3 receptor; range 2.7-6.6More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandPNGBDBM50109477(1-(4-bromophenyl)-3-(2-(furan-2-yl)-8-methyl-8H-py...)
Affinity DataKi:  457nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed