Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50109481'
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50109481BDBM50109481(MRE 3055F20 | 1-(2-furan-2-yl-8-propyl-8H-pyrazolo...)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]MRE 3008F20 from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50109481BDBM50109481(MRE 3055F20 | 1-(2-furan-2-yl-8-propyl-8H-pyrazolo...)
Affinity DataKi:  0.150nMAssay Description:Binding affinity for human adenosine A3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50109481BDBM50109481(MRE 3055F20 | 1-(2-furan-2-yl-8-propyl-8H-pyrazolo...)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]NECA from human adenosine A3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50109481BDBM50109481(MRE 3055F20 | 1-(2-furan-2-yl-8-propyl-8H-pyrazolo...)
Affinity DataKi:  0.150nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/4/2011
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50109481BDBM50109481(MRE 3055F20 | 1-(2-furan-2-yl-8-propyl-8H-pyrazolo...)
Affinity DataKi:  0.150nMAssay Description:Displacement of [3H]MRE3008-F20 from human Adenosine A3 receptor expressed in HEK cells; range 0.10-0.18More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50109481BDBM50109481(MRE 3055F20 | 1-(2-furan-2-yl-8-propyl-8H-pyrazolo...)
Affinity DataKi:  0.530nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50109481BDBM50109481(MRE 3055F20 | 1-(2-furan-2-yl-8-propyl-8H-pyrazolo...)
In Depth
Date in BDB:
5/3/2012
Entry Details Article
PubMed
TargetAdenosine receptor A3(Human)
Università

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50109481BDBM50109481(MRE 3055F20 | 1-(2-furan-2-yl-8-propyl-8H-pyrazolo...)
Affinity DataKi:  151nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/22/2013
Entry Details Article
PubMed