Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with Target = 'Adenosine receptor A3' and Ligand = 'BDBM50550814'
TargetAdenosine receptor A3(Homo sapiens (Human))
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50550814(CHEMBL4747947)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]PSB-11 from human adenosine receptor A3 expressed in CHO cell membranes incubated for 60 mins by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50550814(CHEMBL4747947)
Affinity DataKi:  607nMAssay Description:Displacement of [3H]NECA from rat adenosine receptor A3 expressed in CHO cell membranes incubated for 60 mins by radioligand competition assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50550814(CHEMBL4747947)
Affinity DataEC50:  57nMAssay Description:Antagonist activity at rat A3AR expressed in CHO cells assessed as reduction in NECA-induced inhibition of forskolin-stimulated cAMP accumulation at ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50550814(CHEMBL4747947)
Affinity DataEC50:  1.72E+3nMAssay Description:Antagonist activity at rat A3AR expressed in CHO cells assessed as reduction in NECA-induced inhibition of forskolin-stimulated cAMP accumulation at ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
University of Bonn

Curated by ChEMBL
LigandPNGBDBM50550814(CHEMBL4747947)
Affinity DataEC50:  5.30nMAssay Description:Antagonist activity at rat A3AR expressed in CHO cells assessed as reduction in NECA-induced inhibition of forskolin-stimulated cAMP accumulation inc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed