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Found 7 Enz. Inhib. hit(s) with Target = 'Alpha-1A adrenergic receptor' and Ligand = 'BDBM50118705'
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataKi:  135nMAssay Description:Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataKi:  135nMAssay Description:In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataKi:  140nMAssay Description:Binding affinity towards rat submaxillary gland Alpha-1 adrenergic receptor ; value ranges from (0.12 - 0.15)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataEC50:  603nMAssay Description:Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethraMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataEC50:  60nMAssay Description:Agonist activity at rabbit urethra adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataEC50:  600nMAssay Description:Effective concentration of the compound was determined in vitro against rabbit urethra Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human cloned adrenergic alpha-1A receptor expressed in CHO cells assessed as calcium mobilization by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed