Found 6 Enz. Inhib. hit(s) with Target = 'Amine oxidase [flavin-containing] A' and Ligand = 'BDBM50018671'
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibition of MAO-A in rat liver homogenate preincubated for 240 minsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of MAO-A in rat liver homogenate preincubated for 60 minsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibition of MAO-A in rat liver homogenate preincubated for 30 minsMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of MAO-A in rat liver homogenate using [14C]-5HT as substrate preincubated for 30 mins followed by substrate addition measured after 20 mi...More data for this Ligand-Target Pair
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of human recombinant MAOA using p-tyramine as substrate preincubated for 30 mins followed by substrate addition measured for 1 hr by horse...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Rattus norvegicus (rat))
Okayama University
Curated by ChEMBL
Okayama University
Curated by ChEMBL
Affinity DataIC50: 2.91E+4nMAssay Description:Inhibition of MAO-A in rat liver homogenateMore data for this Ligand-Target Pair