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Found 7 Enz. Inhib. hit(s) with Target = 'Amine oxidase [flavin-containing] A' and Ligand = 'BDBM50197875'
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50197875(CHEMBL3910142)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human recombinant MAOA using p-tyramine as substrate preincubated for 240 mins followed by substrate addition measured for 1 hr by hors...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50197875(CHEMBL3910142)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of human recombinant MAOA using p-tyramine as substrate preincubated for 180 mins followed by substrate addition measured for 1 hr by hors...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50197875(CHEMBL3910142)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of human recombinant MAOA using p-tyramine as substrate preincubated for 120 mins followed by substrate addition measured for 1 hr by hors...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50197875(CHEMBL3910142)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of human recombinant MAOA using p-tyramine as substrate preincubated for 60 mins followed by substrate addition measured for 1 hr by horse...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50197875(CHEMBL3910142)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of human recombinant MAOA using p-tyramine as substrate preincubated for 30 mins followed by substrate addition measured for 1 hr by horse...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50197875(CHEMBL3910142)
Affinity DataIC50:  2.08E+4nMAssay Description:Inhibition of human recombinant MAOA using p-tyramine as substrate preincubated for 15 mins followed by substrate addition measured for 1 hr by horse...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50197875(CHEMBL3910142)
Affinity DataIC50:  1.87E+5nMAssay Description:Inhibition of human recombinant MAOA using p-tyramine as substrate measured for 1 hr by horse-radish peroxidase/amplex red-based fluorometric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed